首页> 外国专利> USE OF 6-SUBSTITUTED 2-QUINOLINONES AND 2-QUINOXALINONES IN THE MANUFACTURE OF MEDICAMENTS FOR CHEMOSENSITIZATION OR RADIOSENSITIZATION, SOME SUCH NEW COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM

USE OF 6-SUBSTITUTED 2-QUINOLINONES AND 2-QUINOXALINONES IN THE MANUFACTURE OF MEDICAMENTS FOR CHEMOSENSITIZATION OR RADIOSENSITIZATION, SOME SUCH NEW COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM

机译:在化学增敏或放射增敏的药物,某些新化合物,其制备方法和组成它们的药物组合物中,使用6-取代的2-喹诺酮和2-喹诺酮类药物

摘要

The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein n, R1, R2, R3, R4 and X have defined meanings.
机译:本发明提供式(I)的化合物,其用作PARP抑制剂的用途以及包含所述式(I)的化合物的药物组合物,其中n,R 1,R 2,R 3,R 4和X具有定义的含义。

著录项

  • 公开/公告号IL176060A

    专利类型

  • 公开/公告日2012-10-31

    原文格式PDF

  • 申请/专利权人 JANSSEN PHARMACEUTICA N.V.;

    申请/专利号IL20060176060

  • 发明设计人

    申请日2006-05-31

  • 分类号C07D241/44;C07D401/12;C07D407/06;C07D409/14;

  • 国家 IL

  • 入库时间 2022-08-21 17:24:47

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