首页> 外国专利> GASTRORESISTANT PHARMACEUTICAL DOSAGE FORM COMPRISING N-(2-(2-PHTHALIMIDOETHOXY)-ACETYL)-L-ALANYL-D-GLUTAMIC ACID (LK-423)

GASTRORESISTANT PHARMACEUTICAL DOSAGE FORM COMPRISING N-(2-(2-PHTHALIMIDOETHOXY)-ACETYL)-L-ALANYL-D-GLUTAMIC ACID (LK-423)

机译:包含N-(2-(2-邻苯二甲氧基)-乙酰基)-L-丙氨酰-D-谷氨酸的耐胃酸药物剂型(LK-423)

摘要

THE PRESENT INVENTION RELATES TO THE PHARMACEUTICAL DOSAGE FORMS WHICH ENABLE A CONTROLLED AND/OR A TARGETED DELIVERY OF AN ACTIVE SUBSTANCE TO THE SELECTED REGIONS OF GASTROINTESTINAL TRACT OF HUMANS OR ANIMALS. THE PHARMACEUTICAL DOSAGE FORMS PREFERABLY COMPRISES THE ACTIVE SUBSTANCE N-(2- (2-PHTHALIMIDOETHOXY)-ACETYL)-L-ALANYL-D-GLUTAMIC ACID (DESIGNATED AS LK 423). METHODS OF TREATMENT OF CHRONIC INFLAMMATORY DISEASES OF GASTROINTESTINAL TRACT OF HUMANS AND / OR ANIMALS BY USING THE PHARMACEUTICAL DOSAGE FORMS OF THE INVENTION ARE DISCLOSED.
机译:本发明涉及可控制地和/或有针对性地将活性物质递送到人或动物胃肠道的选定区域的药物剂量形式。药物剂量形式优选包含活性物质N-(2-(2-邻苯二甲氧基)-乙酰基)-L-丙氨酰-D-谷氨酸(表示为LK 423)。公开了通过使用本发明的药物剂量形式治疗人类和/或动物的胃肠道疾病的慢性炎性疾病的方法。

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