首页> 外国专利> TOPICAL ANTIACNE PREPARATIONS CONTAINING RETINOID (TAZAROTENE OR ADAPALENE), ANTIBIOTIC (CLINDAMYCIN PHOSPHATE) AND/OR KERATOLYTIC (MISCROSPONGED BENZOYL PEROXIDE)

TOPICAL ANTIACNE PREPARATIONS CONTAINING RETINOID (TAZAROTENE OR ADAPALENE), ANTIBIOTIC (CLINDAMYCIN PHOSPHATE) AND/OR KERATOLYTIC (MISCROSPONGED BENZOYL PEROXIDE)

机译:包含视黄醛(塔扎罗汀或阿达帕林),抗菌剂(克林霉素磷酸酯)和/或核解酶(错配过氧化苯甲酰过氧化物)的抗氧化剂

摘要

The present invention relates to a topical preparation for treating acne in the form of a gel and cream comprising Retinoid (Tazarotene or Adapalene) Antibiotic (Clindamycin Phosphate) and/or Keratolytic (Benzoyl Peroxide in microsponges) as active ingredients and a carrier formulated with all or some of the following components: Polyoxyl 35 castor oil Propylene glycol Glycerine, Carbomer, Triethanolamine, EDTA, Emulsifying nonionic wax (Polawax) Ethanol Antioxidants and Preservatives. The present invention advantages regarding state of the art compositions are based on the fact that the present antiacne composition contains a Retinoid, and Antibiotic and/or a Keratolytic agent which allow the control of every kind of acne from mild to vulgar offering less adverse effects.
机译:本发明涉及用于治疗痤疮的凝胶和乳膏形式的局部制剂,其包含类视黄醇(他扎罗汀或阿达帕林)抗生素(克林霉素磷酸酯)和/或角质分解剂(微皂中的过氧化苯甲酰)作为活性成分,以及用所有这些成分配制的载体或以下某些成分:聚氧35蓖麻油丙二醇,甘油,卡波姆,三乙醇胺,EDTA,乳化非离子蜡(Polawax)乙醇抗氧化剂和防腐剂。本发明关于现有技术组合物的优点是基于这样的事实,即本发明的抗痤疮组合物包含类视黄醇,抗生素和/或角质分解剂,该类维生素和/或角质溶解剂可以控制从轻度到普通的各种痤疮,副作用较小。

著录项

  • 公开/公告号EP2049068B1

    专利类型

  • 公开/公告日2011-11-23

    原文格式PDF

  • 申请/专利权人 LABORATORIOS DERMATOLOGICOS DARIER S.A. DE C.V.;

    申请/专利号EP20070789585

  • 发明设计人 AHUMADA AYALA FERNANDO;

    申请日2007-07-25

  • 分类号A61K8/02;A61K8/31;A61K8/34;A61K8/38;A61K8/41;A61K8/44;A61K8/60;

  • 国家 EP

  • 入库时间 2022-08-21 17:16:42

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