首页> 外国专利> IMIDAZOLE-BASED ALKALOID DERIVATIVES WHICH HAVE ANGIOGENESIS INHIBITION AND ANTIOXIDANT EFFECTS AND PRODUCTION METHOD THEREOF

IMIDAZOLE-BASED ALKALOID DERIVATIVES WHICH HAVE ANGIOGENESIS INHIBITION AND ANTIOXIDANT EFFECTS AND PRODUCTION METHOD THEREOF

机译:具有咪唑作用的血管生成抑制和抗氧化剂作用的碱衍生物及其生产方法

摘要

The present invention relates to imidazole-based alkaloid derivatives represented by formula (1) in the description, pharmaceutically acceptable salts, hydrates, solvates, isomers, prodrugs and a preparation method, thereof, and a pharmaceutical composition containing same which has angiogenesis inhibition and antioxidant effects. In the formula, L, M, m, X, Y, R1 and R2 are as defined in the description.
机译:本发明涉及说明书中由式(1)表示的基于咪唑的生物碱衍生物,药学上可接受的盐,水合物,溶剂化物,异构体,前药及其制备方法,以及包含其的具有血管生成抑制作用和抗氧化剂的药物组合物效果。式中,L,M,m,X,Y,R 1和R 2如说明书中所定义。

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