首页> 外国专利> PRE-FREEZE DRIED AZACITIDINE PREPARATION, FREEZE DRIED AZACITIDINE PREPARATION AND METHOD OF MANUFACTURING THE SAME

PRE-FREEZE DRIED AZACITIDINE PREPARATION, FREEZE DRIED AZACITIDINE PREPARATION AND METHOD OF MANUFACTURING THE SAME

机译:冷冻干燥的阿扎替丁制剂,冷冻干燥的阿扎替丁制剂及其制造方法

摘要

The present invention provides a pre-freeze dried azacitidine preparation, a freeze dried azacitidine preparation, and a method of manufacturing the freeze dried azacitidine preparation. The pre-freeze dried azacitidine preparation of the present invention has improved stability in an aqueous solution. When the pre-freeze dried azacitidine preparation is frozen and dried under predetermined process conditions including a freeze drying cycle, a stability-improved freeze dried azacitidine preparation can be usefully produced.
机译:本发明提供了一种预冷冻干燥的阿扎胞苷制剂,一种冷冻干燥的阿扎胞苷制剂以及一种制造该冷冻干燥的阿扎胞苷制剂的方法。本发明的预冻干的阿扎胞苷制剂在水溶液中具有改善的稳定性。当将预冷冻干燥的阿扎胞苷制剂冷冻并在包括冷冻干燥循环的预定工艺条件下干燥时,可以有效地制备稳定性提高的冷冻干燥的阿扎胞苷制剂。

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