首页> 外国专利> A NOVEL AND HIGHLY STEREOSELECTIVE PROCESS FOR PREPARING GEMCITABINE AND INTERMEDIATES THEREOF

A NOVEL AND HIGHLY STEREOSELECTIVE PROCESS FOR PREPARING GEMCITABINE AND INTERMEDIATES THEREOF

机译:一种新型和高度立体选择性的制备吉西他滨及其中间体的方法

摘要

The present invention provides a novel and highly stereoselective process for preparing gemcitabine, which is suitable for industrial production, wherein, it includes the following reactions. Additionally, the invention discloses the key intermediates. The definition for the groups of G1, G2, G3, G4, and G5 are described in the specification.
机译:本发明提供了一种新的且高度立体选择性的制备吉西他滨的方法,其适于工业生产,其中,它包括以下反应。另外,本发明公开了关键中间体。 G1,G2,G3,G4和G5组的定义在说明书中进行了描述。

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