首页> 外国专利> Derivatives (1-4-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-p p p p p p p p p p p p p p p p-2-pi p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p-2-pip p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p_ delta e u a o a o l 1 pain treatment.

Derivatives (1-4-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-pi-p p p p p p p p p p p p p p p p-2-pi p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p-2-pip p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p p_ delta e u a o a o l 1 pain treatment.

机译:衍生物(1-4-π-π-π-π-π-π-π-π-π-π-π-π-PIP pppppppppppppp P-2-πppppppppppppppppppppp ppppppppppp P-2-PIP ppppppppppppppppppppp ppppppppppppppppppppp ppppppppppppppppppppp ppppppppppppppppppppp pppppppp p_ delta euaoaol 1疼痛治疗。

摘要

An object of the present invention is to provide analgesic, anti-inflammatory, diuretic, narcotic, and as a factor of__________for useful compounds. DES, anti-hypertension, anti-alpha-gamma___uuuuuuuuuuuuuuuuuuuuuuuuuuuuuuuuu As a modulator, we learn and memorize the alpha Sigu tau.Neurotransmitters and hormones released as modulators, regulators of renal function, antidepressants, and loss of therapeutic properties Deprivation of memory due to Alzheimer's disease or other alpha__, as an antiepileptic, anticonvulsant, as a therapeutic agent, alcohol, and addictive substance; For controlling the water balance,To control the factors of sodium excretion disorder, to control blood pressure and administration method. (2). The compounds of the present invention are one or more____delta_receptors (ORL-1, mu, delta, kappa) formed by useful pharmacodynamic reactions. (U), R, P, P, or P.The response of the association can be attributed to stimulation (agonist) or inhibition (one or more receptor antagonists). Some compounds can stimulate (for example, a mu agonist) and pause (for example, a different receptor antagonist ORL-1).
机译:本发明的一个目的是提供止痛药,消炎药,利尿药,麻醉药以及有用的化合物的诱因。 DES,抗高血压,抗α-γ___ uuuuuuuuuuuuuuuuuuuuuuuuuuuuuuuuuuu作为调节剂,我们学习并记住αSigu tau。神经递质和激素作为调节剂释放,肾功能调节剂,抗抑郁药,因阿尔茨海默氏病而丧失记忆力和治疗特性丧失或其他alpha__,作为抗癫痫药,抗惊厥药,治疗剂,酒精和成瘾性物质;为了控制水的平衡,控制钠排泄障碍的因素,控制血压和给药方法。 (2)。本发明的化合物是通过有用的药效反应形成的一种或多种δ受体(ORL-1,μ,δ,κ)。 (U),R,P,P或P。关联的响应可归因于刺激(激动剂)或抑制(一种或多种受体拮抗剂)。一些化合物可以刺激(例如,μ激动剂)和停顿(例如,不同的受体拮抗剂ORL-1)。

著录项

  • 公开/公告号CY1109053T1

    专利类型

  • 公开/公告日2014-07-02

    原文格式PDF

  • 申请/专利权人 EURO-CELTIQUE S.A.;

    申请/专利号CY200911000475T

  • 申请日2009-04-29

  • 分类号C07D211/04;A61K31/415;A61K31/4184;A61K31/44;A61K31/445;A61K31/454;A61K31/48;A61P3/04;A61P7/10;A61P9;A61P9/12;A61P11/06;A61P11/10;A61P11/14;A61P13/02;A61P21/02;A61P23;A61P25;A61P25/02;A61P25/04;A61P25/08;A61P25/14;A61P25/22;A61P25/28;A61P25/32;A61P25/36;A61P27/16;A61P29;A61P43;C07D209/34;C07D211/06;C07D235/24;C07D235/26;C07D263/58;C07D401/04;C07D401/06;C07D403/04;C07D403/06;C07D405/14;C07D413/04;C07D413/14;C07D471/04;

  • 国家 CY

  • 入库时间 2022-08-21 15:58:22

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