首页> 外国专利> COMBINATION OF ALPHA-7 ACTIVATORS OF NICOTINE ACETYL-CHOLINE RECEPTOR AND ANTAGONISTS mGluR5, INTENDED FOR APPLICATION FOR DOPKINOM-CAUSED DYSKINESIA, ASSOCIATED WITH CAROSTERN DISEASE

COMBINATION OF ALPHA-7 ACTIVATORS OF NICOTINE ACETYL-CHOLINE RECEPTOR AND ANTAGONISTS mGluR5, INTENDED FOR APPLICATION FOR DOPKINOM-CAUSED DYSKINESIA, ASSOCIATED WITH CAROSTERN DISEASE

机译:烟碱乙酰胆碱受体α-7活化剂和拮抗剂mGluR5的组合,旨在用于因多巴胺引起的运动障碍,与胡萝卜素疾病相关

摘要

The invention relates to new combinations applicable for the treatment of dyskinesia associated with the treatment of Parkinson's disease with a dopamine agonist, comprising as active ingredients at least one low molecular weight activator of the nicotinic acetylcholine receptor alpha-7 and at least one low molecular weight metabotropic antagonist glutamate receptor 5; to receive them; to their use as medicines and to medicines containing them.
机译:本发明涉及适用于用多巴胺激动剂治疗与帕金森氏病相关的运动障碍的新组合,其包含至少一种烟碱型乙酰胆碱受体α-7的低分子量活化剂和至少一种低分子量作为活性成分。代谢型拮抗剂谷氨酸受体5;接收它们;用作药物或含有它们的药物。

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