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MONOCYCLIC AND BICYCLIC HIMBACINE DERIVATIVES USEFUL AS THROMBIN RECEPTOR ANTAGONISTS
MONOCYCLIC AND BICYCLIC HIMBACINE DERIVATIVES USEFUL AS THROMBIN RECEPTOR ANTAGONISTS
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机译:用作凝血酶受体拮抗剂的单环和双环联苯胺衍生物
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摘要
Monocyclic and bicyclic himbacine derivatives of the formula or a pharmaceutically acceptable salt or solvate of said compound wherein represents an optional double bond and wherein Gn, Jn, R3, R8, R9, R10, R11, R32, R33, B and Het are herein defined are disclosed, as well as pharmaceutical compositions containing them and a method of treating diseases associated with thrombosis, atherosclerosis, restenosis, hypertension, angina pectoris, arrhythmia, heart failure, and cancer by administering said compounds. Combination therapy with other agents is also claimed.
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