首页> 外国专利> Crystalline forms of N- (tert-butoxycarbonyl) -3-methyl-L-valyl- (4R) -4 - ((7-chloro-4-methoxy-1-isoquinolinyl) oxy) -N - ((1R, 2S) -1 - ((cyclopropylsulfonyl) carbamoyl) -2-vinylcyclopropyl) -L-prolinamide

Crystalline forms of N- (tert-butoxycarbonyl) -3-methyl-L-valyl- (4R) -4 - ((7-chloro-4-methoxy-1-isoquinolinyl) oxy) -N - ((1R, 2S) -1 - ((cyclopropylsulfonyl) carbamoyl) -2-vinylcyclopropyl) -L-prolinamide

机译:N-(叔丁氧羰基)-3-甲基-L-戊基-(4R)-4-((7-氯-4-甲氧基-1-异喹啉基)氧基)-N-((1R,2S)的晶体形式-1-(((环丙基磺酰基)氨基甲酰基)-2-乙烯基环丙基)-L-脯氨酰胺

摘要

The present disclosure generally relates to crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N-((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide. The present disclosure also generally relates to a pharmaceutical composition comprising one or more of the crystalline forms, as well as methods of using the crystalline forms in the treatment of Hepatitis C virus (HCV) and methods for obtaining such crystalline forms.
机译:本公开总体上涉及N-(叔丁氧基羰基)-3-甲基-L-戊基-(4R)-4-(((7-氯-4-甲氧基-1-异喹啉基)氧基)-N-的晶体形式。 (((1R,2S)-1-((环丙基磺酰基)氨基甲酰基)-2-乙烯基环丙基)-L-脯氨酰胺。本公开内容还总体上涉及包含一种或多种晶型的药物组合物,以及在治疗丙型肝炎病毒(HCV)中使用晶型的方法和获得这种晶型的方法。

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