首页> 外国专利> NEW CRYSTALLINE POLYMORPHIC FORMS OF HEMINAPADHYSILATE 5- (2 - {6- (2,2-DIFFOR-2-PHENYLETOXI) HEXIL AMINO} -1- (R) -HYDROXIETHYL) -8-HYDROXYCHINOHLON-NY-HON-3- (R) -HYDROXYETHYL)) -1- (R) -HYDROXYETHYL)) -1- (R) -HYDROXYETHYLY The quality of β-adrenergic receptor agonists

NEW CRYSTALLINE POLYMORPHIC FORMS OF HEMINAPADHYSILATE 5- (2 - {6- (2,2-DIFFOR-2-PHENYLETOXI) HEXIL AMINO} -1- (R) -HYDROXIETHYL) -8-HYDROXYCHINOHLON-NY-HON-3- (R) -HYDROXYETHYL)) -1- (R) -HYDROXYETHYL)) -1- (R) -HYDROXYETHYLY The quality of β-adrenergic receptor agonists

机译:氨甲酰5-(2--[[[6-(2,2-DIFFOR-2-苯氧基)己基]氨基] -1-(R)-羟乙基)-8-羟基甲壳素-NY-HON-3-的结晶多态新形式(R)-羟乙基))-1-(R)-羟乙基))-1-(R)-羟乙基β-肾上腺素能受体激动剂的质量

摘要

The application describes new crystalline polymorphic forms of the heminapadisylate 5- (2 - {[6- (2,2-difluoro-2-phenylethoxy) hexyl] amino} -1- (R) -hydroxyethyl) -8-hydroxyquinoline-2 (1H) -she. The application also describes pharmaceutical compositions containing these crystalline polymorphic forms, methods for their use in the treatment of respiratory diseases associated with β2 adrenergic receptor activity, and a method for producing such crystalline polymorphic.
机译:该申请描述了半乙酰二甲酸酯5-(2-{[6-(2,2-二氟-2-苯基乙氧基)己基]氨基} -1-(R-羟乙基)-8-羟基喹啉-2( 1H)-她。该申请还描述了包含这些结晶多晶型物形式的药物组合物,其用于治疗与β2肾上腺素能受体活性有关的呼吸道疾病的方法,以及制备这种结晶多晶型物的方法。

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