首页> 外国专利> ACETYLCHOLINESTERASE INHIBITOR COMPOUNDS AND 5HT4 SEROTONERGIC RECEPTOR AGONISTS, WITH PROMNESIA EFFECT, METHODS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

ACETYLCHOLINESTERASE INHIBITOR COMPOUNDS AND 5HT4 SEROTONERGIC RECEPTOR AGONISTS, WITH PROMNESIA EFFECT, METHODS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME

机译:乙炔胆碱酯酶抑制剂化合物和5HT4血清激素受体激动剂,具有预后效应,其制备方法和包含相同成分的药物成分

摘要

The invention relates to compounds of formula (I) as well as to neurogenic enantiomers thereof, acid salts thereof, hydrates thereof or to solvation products thereof. Among a large number of possible meanings, X is a halogen, Y is an oxygen atom; all the coefficients m, n, r and s have a value of 1, R is a methyl, and R' is a cycloalkyl. The invention also includes methods for preparing the above compounds and pharmaceutical compositions including same.
机译:本发明涉及式(I)化合物及其神经原性对映异构体,其酸盐,其水合物或其溶剂化产物。在许多可能的含义中,X是卤素,Y是氧原子;所有系数m,n,r和s的值为1,R为甲基,R'为环烷基。本发明还包括制备上述化合物的方法和包括该化合物的药物组合物。

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