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Pest Control Agents for parasitic Honey Bee pests and Pest Control method for parasitic Honey Bee pests through the use of Pest Control agents

机译:通过使用害虫防治剂防治蜜蜂寄生虫的病虫害防治方法和方法

摘要

With a high degree of Security for honey bees and that shows excellent control effects against pests parasitic Pest of Honey bees.Claim 1: an agent control pests parasitic Honeybees, characterized in that it comprises: at least a compound represented by the formula (1) or acid Addition salts of that as an active ingredient, (in the formula (1), ar represents a phenyl Group can be Substituted Heterocycles, a 5 to 6 members can be replaced,Heterocicloalquilo or a group of 4 to 10 members; a represents a Heterocyclic 5 to 10 members has a Link that includes one or more unsaturated nitrogen ATOMS, and a group that is replaced with an imino Group r in a position adjacent to the nitrogen Atom in the cicl Or; and represents a hydrogen Atom, a Halogen Atom, hydroxyl Group,A cu2081u208bu2086 alkyl group can be substituted with a Halogen Atom, a Group cu2081u208bu2086 alquiloxi can be substituted with a Halogen Atom or a cyano Group, a Nitro Group; and R represents any Remnants of the Group represented by the formula (2), here, ru00b9 represents A Hydrogen Atom, an alkyl group cu2081u208bu2086 replaced,A Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, or a group pentafluorofenilo; Ru00b2 represents an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Group cu2083 u208bu2086 branched alkyl substituted cyclic or not, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a substituted or unsubstituted aryl Group cu2086u208bu2081u2080, 5 to 10 members heterocycle substituted or unsubstituted benzyl group or a substituted or unsubstituted; ru00b3 represents an alkyl group which may cu2081u208bu2086 Replace with a Halogen Atom, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a Group cu2086u208bu2081u2080 aryl substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2081u208bu2086 alkyl substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo replaced or not replaced, a group Cu2086u208bu2081u2080 or aryl - substituted or non substituted cu2082u208bu2086 alquinilo cu2081u208bu2086 alkyl phenoxy Group, a substituted or unsubstituted,A Group cu2082u208bu2086 alquenilo phenoxy substituted or non substituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo, a 5 to 10 members heterocycle substituted or unsubstituted heterocycle - a group of 5 to 10 members cu2081u208bu2086 alkyl substituted or non substituted Heterocyclic Group, a - cu2082u208bu2086 alquenilo 5-10 members replaced or not replacedA Group cu2082u208bu2086 alquinilo heterocycle - 5 to 10 members replaced or not replaced, a Group cu2081u208bu2084 cu2081u208bu2085 - alkoxy alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 cu2082u208bu2085 alquinilo alkoxy -, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a cu2081 u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo or a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo; ru2074 represents a hydrogen Atom, a group Formilo,A cu2081u208bu2081u2088 alkyl group can be replaced, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a substituted or unsubstituted aryl Group cu2086u208bu2081u2080, a Group cu2086u208bu2081u2080 ar ILO cu2081u208bu2086 alkyl substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo replaced or not replacedA Group cu2086u208bu2081u2080 aryl - substituted or non substituted cu2082u208bu2086 alquinilo cu2081u208bu2086 alkyl phenoxy Group, a substituted or unsubstituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquenilo phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo heterocycle, a 5 to 10 Wed E substituted or unsubstituted heterocycle cu2081u208bu2086 alkyl -, a group of 5 to 10 members replaced or not replacedA Group cu2082u208bu2086 alquenilo heterocycle - 5 to 10 members substituted or unsubstituted heterocycle cu2082u208bu2086 alquinilo - a group of 5 to 10 members replaced or not replaced, a Group cu2081u208bu2084 cu2081u208bu2085 - alkoxy alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 alcox I cu2082u208bu2085 alquinilo, a cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo,Or a group represented by the remains of a group of formulas (3) here, ru2074u1d43, ru2074u1d47 and ru2074u1d9c represent an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquini It can be substituted with a Halogen Atom, a substituted or unsubstituted aryl Group cu2086u208bu2081u2080,A Group cu2086u208bu2081u2080 cu2081u208bu2086 alkyl aryl - substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquinilo substituted or unsubstituted phenoxy cu2081u208bu2086 alkyl group, a substituted or non substituted a g He cu2082u208bu2086 alquenilo phenoxy substituted or non substituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo,A 5 to 10 members heterocycle substituted or non substituted Heterocyclic Group, a - 5 to 10 members cu2081u208bu2086 alkyl substituted or non substituted Heterocyclic Group, a - cu2082u208bu2086 alquenilo 5-10 members substituted or unsubstituted heterocycle cu2082u208bu2086 alquinilo - a group of 5 to 10 members Substituted or non substituted alkoxy -, a Group cu2081u208bu2084 cu2081u208bu2085 alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo,A Group cu2081u208bu2084 cu2082u208bu2085 alquinilo alkoxy -, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo or a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo, ru2074u1d48 represents an alkyl group cu2081u208bu2086 can be replaced with an atom of halu00f3gen Or, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom,A cu2086u208bu2081u2080 aryl group or a substituted or non substituted heterocycle of 5-10 members replaced or not replaced, and ru2074u1d49 and ru2074u1da0 represent each independently a hydrogen Atom, an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Group cu2082 u208bu2086 alquenilo can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a cu2086u208bu2081u2080 aryl group or a substituted or non substituted heterocycle of 5-10 members replaced or not replaced; ru2075 represents an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Cu2082u208bu2086 alquenilo Group can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a Group cu2086u208bu2081u2080 aryl substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2081u208bu2086 alkyl substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo replaced or not replaced, a group Cu2086u208bu2081u2080 or aryl - substituted or non substituted cu2082u208bu2086 alquinilo cu2081u208bu2086 alkyl phenoxy Group, a substituted or unsubstituted,A Group cu2082u208bu2086 alquenilo phenoxy substituted or non substituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo, a 5 to 10 members heterocycle substituted or unsubstituted heterocycle - a group of 5 to 10 members cu2081u208bu2086 alkyl substituted or non substituted Heterocyclic Group, a - cu2082u208bu2086 alquenilo 5-10 members replaced or not replacedA Group cu2082u208bu2086 alquinilo heterocycle - 5 to 10 members replaced or not replaced, a Group cu2081u208bu2084 cu2081u208bu2085 - alkoxy alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 cu2082u208bu2085 alquinilo alkoxy -, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a cu2081 u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo or a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo; ru2076 represents a hydrogen Atom, a group Formilo, a phosphoryl group or- cu2081u208bu2084 alkyl or alkyl group, a cu2081u208bu2081u2088 can be replaced, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a substituted or unsubstituted aryl Group cu2086u208bu2081u2080, a - cu2081u208bu2086 alkyl aryl Group cu2086u208bu2081u2080 replaced or not replaced, a Group cu2086u208bu2081u2080 aryl - cu2082u208bu2086 alquenilo replaced or not replacedA Group cu2086u208bu2081u2080 aryl - substituted or non substituted cu2082u208bu2086 alquinilo cu2081u208bu2086 alkyl phenoxy Group, a substituted or unsubstituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquenilo phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo heterocycle, a 5 to 10 Wed E substituted or unsubstituted heterocycle cu2081u208bu2086 alkyl -, a group of 5 to 10 members replaced or not replacedA Group cu2082u208bu2086 alquenilo heterocycle - 5 to 10 members substituted or unsubstituted heterocycle cu2082u208bu2086 alquinilo - a group of 5 to 10 members replaced or not replaced, a Group cu2081u208bu2084 cu2081u208bu2085 - alkoxy alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 alcox I cu2082u208bu2085 alquinilo, a cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo,Or a group represented by the remains of a group of formulas (4) here, ru2076u1d43, ru2076u1d47 and ru2076u1d9c represent an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquini It can be substituted with a Halogen Atom, a substituted or unsubstituted aryl Group cu2086u208bu2081u2080,A Group cu2086u208bu2081u2080 cu2081u208bu2086 alkyl aryl - substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquinilo substituted or unsubstituted phenoxy cu2081u208bu2086 alkyl group, a substituted or non substituted a g He cu2082u208bu2086 alquenilo phenoxy substituted or non substituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo,A 5 to 10 members heterocycle substituted or non substituted Heterocyclic Group, a - 5 to 10 members cu2081u208bu2086 alkyl substituted or non substituted Heterocyclic Group, a - cu2082u208bu2086 alquenilo 5-10 members substituted or unsubstituted heterocycle cu2082u208bu2086 alquinilo - a group of 5 to 10 members Substituted or non substituted alkoxy -, a Group cu2081u208bu2084 cu2081u208bu2085 alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo,A Group cu2081u208bu2084 cu2082u208bu2085 alquinilo alkoxy -, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo or a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo, ru2076u1d48 represents an alkyl group cu2081u208bu2086 can be replaced with an atom of halu00f3gen Or, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom,A cu2086u208bu2081u2080 aryl group or a substituted or non substituted heterocycle of 5-10 members replaced or not replaced, ru2076u1d49 and ru2076u1da0 represent each independently a hydrogen Atom, an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Group cu2082 u208bu2086 alquenilo can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, an alkyl group, alkoxy cu2081u208bu2084 - cu2081u208bu2085, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, an aryl substituted or non substituted cu2086u208bu2081u2080, a Group cu2086u208bu2081u2080 cu2081u208bu2086 alkyl aryl - substituted or not Heterocycle substituted or 5 to 10 members replaced or not replaced, ru2076u1d4d and ru2076u02b0 represent each independently a hydrogen Atom,A cu2081u208bu2086 alkyl group can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, or a Group cu2086u208bu2081u2080 aryl substituted or non substituted A 5 to 10 members heterocycle substituted or non substituted, and ru2076u2071, ru2076u02b2 and ru2076u1d4f represent each independentlyA Hydrogen Atom, an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom or an aryl Group cu2086u208bu2081u2080 their Replaced or not replaced; and ru2077 represents an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a Group cu2086u208bu2081u2080 aryl substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2081u208bu2086 alkyl substituted or non substituted a g He cu2086u208bu2081u2080 aryl - cu2082u208bu2086 alquenilo substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquinilo replaced or not replacedA Group cu2081u208bu2086 alkyl phenoxy substituted or unsubstituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquenilo phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo, a 5 to 10 members heterocycle substituted or non substituted Heterocyclic Group, an alkyl cu2081u208bu2086 - 5 10 members replaced or not replacedA Group cu2082u208bu2086 alquenilo heterocycle - 5 to 10 members substituted or unsubstituted heterocycle cu2082u208bu2086 alquinilo - a group of 5 to 10 members replaced or not replaced, a Group cu2081u208bu2084 cu2081u208bu2085 - alkoxy alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 alcox I cu2082u208bu2085 alquinilo, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkylA Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo or a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo; yu00b9 and yu00b2 represents an oxygen Atom or a Sulfur Atom, and can be the same or different; and ru02b8 represents an alkyl group cu2081u208bu2086 can be replaced with an atom of halu00f3gen Or, a Group cu2082u208bu2086 alquenilo can be substituted with a Halogen Atom,A Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom, a Group cu2086u208bu2081u2080 aryl substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2081u208bu2086 alkyl substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo replaced or not replaced, a group Cu2086u208bu2081u2080 or aryl - substituted or non substituted cu2082u208bu2086 alquinilo cu2081u208bu2086 alkyl phenoxy Group, a substituted or unsubstituted,A Group cu2082u208bu2086 alquenilo phenoxy substituted or non substituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquinilo, a 5 to 10 members heterocycle substituted or unsubstituted heterocycle cu2081u208bu2086 alkyl -, a group of 5 to 10 members replaced or not replacedA Group cu2082u208bu2086 alquenilo heterocycle - 5 to 10 members replaced or not replaced or heterocycle Group - cu2082u208bu2086 alquinilo 5-10 members replaced or not replaced; ru1dbb represents an alkyl group cu2081u208bu2086 can be substituted with a Halogen Atom, a group that cu2082u208bu2086 Nile can be substituted with a Halogen Atom, a Group cu2082u208bu2086 alquinilo can be substituted with a Halogen Atom,A Group cu2086u208bu2081u2080 aryl substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2081u208bu2086 alkyl substituted or non substituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquenilo substituted or unsubstituted aryl Group, a cu2086u208bu2081u2080 - cu2082u208bu2086 alquinilo replaced or not replaced, Group F Enoxi - cu2081u208bu2086 alkyl substituted or non substituted phenoxy Group, a substituted or unsubstituted cu2082u208bu2086 alquenilo,A Group cu2082u208bu2086 alquinilo phenoxy substituted or unsubstituted heterocycle, a 5 to 10 members substituted or unsubstituted heterocycle -, a group of 5 to 10 members cu2081u208bu2086 alkyl substituted or non substituted Heterocyclic Group, a - cu2082u208bu2086 alquenilo 5-10 members replaced or not replaced OJ alquinilo - cu2082u208bu2086 heterocycle, a group of 5 to 10 members replaced or not replacedA Group cu2081u208bu2084 cu2081u208bu2085 - alkoxy alkyl alkoxy -, a Group cu2081u208bu2084 cu2082u208bu2085 alquenilo, a Group cu2081u208bu2084 cu2082u208bu2085 alquinilo alkoxy -, a Group cu2081u208bu2084 Alquiltio - cu2081u208bu2085 alkyl group, a cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquenilo or a Group cu2081u208bu2084 Alquiltio - cu2082u208bu2085 alquinilo; And N represents 1 or 2).
机译:权利要求1:一种防治害虫寄生性蜜蜂的药剂,其特征在于:至少包含一种由式(1)表示的化合物,该蜜蜂对蜜蜂具有很高的安全性,并且对蜜蜂的有害生物具有优异的防治效果。或作为活性成分的酸加成盐(在式(1)中,ar表示苯基可被取代的杂环,可取代5至6个成员,杂cloalquilo或4至10个成员的基团; a表示杂环的5至10个成员具有一个环,该环包括一个或多个不饱和氮原子ATOMS,以及一个在基团Or中与氮原子相邻的位置被亚氨基r取代的亚氨基;并且表示氢原子,卤素原子,羟基,c c 1 2 3烷基可以被卤素原子取代,c 1 2 3基团可以被卤素原子或氰基,硝基取代;以及R代表Grou的任何残余物由式(2)表示的p,其中,r u00b9代表氢原子,烷基被c u2081 u208b u2086取代,A基团c u2082 u208b u2086alquenilo可以被卤素原子取代,a c u2082 u208b u2086组alquinilo可以被卤素原子或五氟fenilo组取代; R u00b2代表烷基c u2081 u208b u2086可以被卤素原子取代,c u2083 u208b u2086支链的烷基取代或不被环状取代,c u2082 u208b u20b的烷基可以是用卤素原子取代,基团c u2082 u208b u2086 alquinilo可以被卤素原子,取代或未取代的芳基c u2086 u208b u2081 u2080取代,具有5至10个杂环取代或未取代的苄基或取代或未取代; r u00b3表示可以被卤素原子取代的烷基,基团c u2082 u208b u2086 alquenilo可以被卤素原子取代,c u2082 u208b u208b u2086 alquinilo可以被卤素原子取代,基团c u2086 u208b u2081 u2080芳基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2081 u208b u2086烷基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u2086 alquenilo已取代或未取代,C u2086 u208b u2081 u2080或芳基-取代或未取代的c u2082 u208b u2086 alquinilo c u2081 u208b u2086烷基苯氧基,取代或未取代的,A c u2082 u208b u2086烷氧基苯氧基取代或未取代的苯氧基,取代或未取代的c u2082 u208b u20b u2086喹啉,5至10个成员的杂环取代或未取代的杂环-5至10个成员的一组c u2081 u208b u2086烷基被取代或未被取代杂环基团-替换或未替换a-c u2082 u208b u2086 alquenilo组c u2082 u208b u2086 alquinilo杂环-替换或未替换5至10个成员,c u2081 u208b u2084组c u2081 u208b u2085-烷氧基烷基烷氧基-,组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u208b u2084 c u2082 u208b u2085烷氧基烷氧基- ,c u2081 u208b u2084 Alquiltio烷基组,ac u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo或c u2081 u208b u2084 Alquiltio组-c u2082 u208b u2085 alquinilo; r u2074代表氢原子,基团为Formilo,一个c u2081 u208b u2081 u2088烷基可被取代,一个c u2082 u208b u2086烷基被卤素原子取代,一个c u2082 u208b u2086 alquinilo可以被卤素原子,取代或未取代的芳基c u2086 u208b u2081 u2080,c u2086 u208b u2081 u2080组和ILO c u2081 u208b u2086取代烷基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u2086 alquenilo取代或未取代A组c u2086 u208b u2081 u2080芳基-取代或未取代的c u2082 u208b u2086 alquinilo c u2081 u208b u2086烷基苯氧基,取代或未取代的苯氧基,取代或未取代的c u2082 u208b u20b Alquenilo苯氧基,取代或未取代的c u2082 u208b u2086 alquinilo杂环,是5到10个Wed E取代或未取代的杂环c u2081 u208b u2086烷基-,一个5到10个成员的组被取代或未取代acedA组c u2082 u208b u2086 Alquenilo杂环-5至10个取代或未取代的杂环c u2082 u208b u2086 alquinilo-一组5至10个成员被取代或未取代,组c u2081 u208b u2084 c u2081 u208b u2085-烷氧基烷基烷氧基-,组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u208b u2084 alcox I c u2082 u208b u2085 alquinilo ,ac u2081 u208b u2084 Alquiltio-c u2081 u208b u2085烷基,组c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo,一组c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquinilo,或由一组公式(3)的残基表示的组,此处为r u2074 u1d43,r u2074 u1d47和r u2074 u1d9c表示烷基c u2081 u208b u2086可以被卤素原子取代,c u2082 u208b u2086烷基可以被卤素原子取代,c u2082 u208b 可以被卤素原子,取代或未取代的芳基c u2086 u208b u2081 u2080,A组c u2086 u208b u2081 u2080 c u2081 u208b u2086烷基芳基取代-或非取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u2086 Alquenilo取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u208b u2086 alquinilo取代或未取代苯氧基c u2081 u208b u2086烷基,取代或未取代的ag He c u2082 u208b u2086 alquenilo苯氧基取代或未取代的苯氧基,取代或未取代的c u2 082 u208b u2086 Alquinilo,5至10个成员的杂环取代或未取代的杂环基,a-5至10个成员c u2081 u208b u2086烷基取代或未取代的杂环基,a-c u2082 u208b u2086 alquenilo 5-10个取代或未取代的杂环c u2082 u208b u2086 alquinilo-一组5至10个取代或未取代的烷氧基-组c u2081 u208b u2084 c u2081 u208b u2085烷基烷氧基-组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u208b u2084 c u2082 u208b u2085 alquinilo烷氧基-组c u2081 u208b u2084 Alquiltio -c u2081 u208b u2085烷基,ac u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo或基团c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquinilo,r u2074 u1d48表示烷基c u2081 u208b u2086可以被hal u00f3gen原子取代,或者c u2082 u208b u2086 alquenilo基团可以被卤素原子取代,c u2082基团 u208 b u2086 alquinilo可以被卤素原子,c u2086 u208b u2081 u2080芳基或5-10个取代或未取代的取代或未取代杂环取代,并且r u2074 u1d49和r u2074 u1da0各自独立地表示氢原子,烷基c u2081 u208b u2086可以被卤素原子取代,c u2082 u208b u2086烷基可以被卤素原子取代,c组u2082 u208b u2086 alquinilo可以被卤素原子,ac u2086 u208b u2081 u2080芳基或5-10个被取代或未被取代的取代或未取代的杂环取代; r u2075表示烷基c u2081 u208b u2086可以被卤素原子取代,C u2082 u208b u2086烷基可以被卤素原子取代,基团c u2082 u208b u20b alquinilo可以被卤素原子取代,基团c u2086 u208b u2081 u2080芳基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2081 u208b u2086烷基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u2086 alquenilo已取代或未取代,C u2086 u208b u2081 u2080或芳基-取代或未取代的c u2082 u208b u2086 alquinilo c u2081 u208b u2086烷基苯氧基,取代或未取代的,A c u2082 u208b u2086烷氧基苯氧基取代或未取代的苯氧基,取代或未取代的c u2082 u208b u20b u2086喹啉,5至10个成员的杂环取代或未取代的杂环-5至10个成员的一组c u2081 u208b u2086烷基被取代或未被取代d杂环基团-a-替换或不替换5-10个成员的c u2082 u208b u2086 alquenilo杂环-替换或不替换的5-10个成员c u2082 u208b u20b的杂环基,c u2081 u208b u2084 c u2081 u208b u2085-烷氧基烷基烷氧基-,组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u208b u2084 c u2082 u208b u2085 alquinilo烷氧基-,一个c u2081 u208b u2084 Alquiltio烷基-ac u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo或c u2081 u208b u2084组Alquiltio-c u2082 u208b u2085 alquinilo; r u2076代表氢原子,基团Formilo,磷酰基或-c u2081 u208b u2084烷基或烷基,可以替换ac u2081 u208b u2081 u2088,基团c u2082 u208b u2086 alquenilo可以被卤素原子取代,基团c u2082 u208b u2086 alquinilo可以被卤素原子,取代或未取代的芳基c u2086 u208b u2081 u2080取代,a-c u2081 u208b u2086烷基芳基c u2086 u208b u2081 u2080组已替换或未替换,c u2086 u208b u2081组uu8080芳基-c u2082 u208b u2086 alquenilo已替换或未替换A组c u2086 u208b u2081 u2080芳基-取代或未取代的c u2082 u208b u2086 Alquinilo c u2081 u208b u2086烷基苯氧基,取代或未取代的苯氧基,取代或未取代的c u2082 u208b u2086烷基苯氧基,取代或未取代的c u2082 u208b u2086 Alquinilo杂环,5到10个Wed E取代或未取代的杂环c u2081 u208b u2086烷基-,一组5到10个成员被替换或未替换A组c u2082 u208b u2086 Alquenilo杂环-5到10个成员被取代或未取代的杂环c u2082 u208b u2086 alquinilo-一组5到10个成员被替换或未替换,组c u2081 u208b u2084 c u2081 u208b u2085-烷氧基烷基烷氧基-,组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u208b u2084 alcox I c u2082 u208b u2085 alquinilo,ac u2081 u208b u2084烷基,基团c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo,一组c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquinilo,或此处为一组公式(4)的残差表示的组r u2076 u1d43,r u2076 u1d47和r u207 6 u1d9c表示烷基c u2081 u208b u2086可以被卤素原子取代,c u2082 u208b u2086烷基可以被卤素原子取代,c u2082 u208b u208b u2086烷基它可以被卤素原子,取代或未取代的芳基c u2086 u208b u2081 u2080取代,A组c u2086 u208b u2081 u2080 c u2081 u208b u2086烷基芳基-取代或未取代芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u20b Alquenilo取代或未取代芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u208b u2086 Alquinilo取代或未取代的苯氧基c u2081 u208b u2086烷基,取代或未取代的ag He c u2082 u208b u208b u20b烷氧基苯氧基取代或未取代的c u2082 u208b u20b u2086烷基,5至10个成员杂环取代或未取代的杂环基,a-5至10个成员c u2081 u208b u2086烷基取代或未取代d杂环基团-a-c u2082 u208b u2086 Alquenilo 5-10个取代或未取代的杂环c u2082 u208b u20b alquinilo-5至10个成员的取代或未取代的烷氧基-组c u2081 u208b u2084 c u2081 u208b u2085烷基烷氧基-,组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,A组c u2081 u208b u2084 c u2082 u208b u2085 alquinilo烷氧基-一组c u2081 u208b u2084 Alquiltio-烷基 ac u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo或一组c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquinilo,r u2076 u1d48表示烷基c u2081 u208b u2086可以被hal u00f3gen原子取代,或组c u2082 u208b u2086 alquenilo可以被卤素原子取代,基团c u2082 u208b u2086 alquinilo可以被卤素原子,c u2086 u208b u2081 u2080芳基或5-10个成员的取代或未取代的杂环取代更换或不更换ed,r u2076 u1d49和r u2076 u1da0各自独立地表示氢原子,烷基c u2081 u208b u2086可以被卤素原子取代,c u2082 u208b u2086基团alquenilo可以是c u2082 u208b u2086 alquinilo组可以被卤素原子取代,烷基,烷氧基,烷氧基c u2081 u208b u2084-c u2081 u208b u2085组c u2081 u208b u2084 Alquiltio-c u2081 u208b u2085烷基,芳基取代或未取代的c u2086 u208b u2081 u2080,基团c u2086 u208b u2081 u2080 c u2081 u208b u2086烷基芳基-取代或未杂环取代或5至10个成员被取代或未被取代,r u2076 u1d4d和r u2076 u02b0各自独立地表示氢原子,c u2081 u208b u2086烷基可被卤素原子,c u2082 u208b u2086组alquenilo可以被卤素原子取代,c u2082 u208b u20b组alquinilo可以被卤素原子或c u2086组208b u2081 u2080芳基取代或未取代的A 5-10元杂环取代或未取代的基团,并且r u2076 u2071,r u2076 u02b2和r u2076 u1d4f各自独立地表示氢原子,烷基c u2081 u208b u2086可以被卤素原子取代,c u2082 u208b u2086组alquenilo可以被卤素原子取代,c u2082 u208b u2086 alquinilo组可以被卤素原子或芳基c u2086 u208b u2081 u2080其已取代或未取代;和r u2077代表烷基c u2081 u208b u2086可以被卤素原子取代,c u2082 u208b u2086组可以被卤素原子取代,c u2082 u208b u2086组alquinilo可以被卤素原子取代,卤素原子是c u2086 u208b u2081 u2080芳基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2081 u208b u2086烷基取代或未取代的ag He c u2086 u208b u2081 u2080芳基-c u2082 u208b u20b Alquenilo取代或未取代的芳基, ac u2086 u208b u2081 u2080-c u2082 u208b u2086取代或未取代的烷基c u2081 u208b u20b烷基苯氧基取代或未取代的苯氧基,取代或未取代的c u2082 u208b u2086 alquenilo苯氧基,取代或未取代的c u2082 u208b u2086 alquinilo,5至10个成员的杂环取代或未取代的杂环基,烷基c u2081 u208b u2086-5个10个被取代或未取代的成员c u2082 u208b u2086 Alquenilo杂环-5至10个取代或未取代的杂环c u2082 u208b u2086 alquinilo-一组5至10个被取代或未取代的成员,一组c u2081 u208b u2084 c u2081 u208b u2085-烷氧基烷基烷氧基-c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u 208b u2084 alcox I c u2082 u208b u2085 alquinilo,组c u2081 u208b u2084 Alquiltio-c u2081 u208b u2085烷基A组c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo或Group c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquinilo; y u00b9和y u00b2代表氧原子或硫原子,可以相同或不同;并且r u02b8表示烷基c u2081 u208b u2086可以被hal u00f3gen原子取代,或者c u2082 u208b u2086 Alquenilo基团可以被卤素原子取代,c u2082基团 u208b u2086 alquinilo可以被卤素原子,c u2086 u208b u2081 u2080芳基取代或未取代的芳基取代,ac u2086 u208b u2081 u2080-c u2081 u208b u2086烷基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u2086 alquenilo取代或未取代,基团C u2086 u208b u2081 u2080或芳基-取代或未取代的c u2082取代基或未取代的烷基苯氧基,取代基或未取代的烷基苯氧基,取代基或未取代的烷基,取代基或未取代基alquinilo,一个5至10个成员的杂环取代或未取代的杂环c u2081 u208b u2086烷基-,一个5至10个成员被取代或未被取代的基团replaceA组c u2082 u208b u2086 alquenilo杂环-5至10个成员已被替换或未替换,或杂环组-c u2082 u208b u20b alquinilo有5-10个成员已被替换或未替换; r u1dbb代表烷基c u2081 u208b u2086可被卤素原子取代,c u2082 u208b u2086尼罗尔可被卤素原子取代,基团c u2082 u208b u2086 alquinilo可以被卤素原子取代,c u2086 u208b u2081 u2080芳基取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2081 u208b u20b烷基取代或未取代芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u2086 Alquenilo取代或未取代的芳基,ac u2086 u208b u2081 u2080-c u2082 u208b u208b u2086 alquinilo已取代或未取代, F群Enoxi-c u2081 u208b u2086烷基取代或未取代的苯氧基,取代或未取代的c u2082 u208b u2086烷基,A组c u2082 u208b u2086萘基苯氧基取代或未取代的杂环,a 5到10个取代或未取代的杂环--5至10个成员的c u2081 u208b u2086烷基被取代或未被取代杂环基团-a-c u2082 u208b u2086 alquenilo 5-10个成员被替换或未替换OJ alquinilo-c u2082 u208b u20b杂环,一组5至10个成员被替换或未替换A组c u2081 u208b u2084 c u2081 u208b u2085-烷氧基烷基烷氧基-,组c u2081 u208b u2084 c u2082 u208b u2085 alquenilo,组c u2081 u208b u2084 c u2082 u208b u2085 alquinilo烷氧基-一组c u2081 u208b u2084 Alquiltio烷基,ac u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquenilo或一组c u2081 u208b u2084 Alquiltio-c u2082 u208b u2085 alquinilo; N代表1或2)。

著录项

  • 公开/公告号AR098538A1

    专利类型

  • 公开/公告日2016-06-01

    原文格式PDF

  • 申请/专利权人 MEIJI SEIKA PHARMA CO. LTD.;

    申请/专利号AR2014P104425

  • 发明设计人

    申请日2014-11-26

  • 分类号C07D401/06;A01N43/40;A01N43/42;A01N43/54;A01N43/58;A01N43/60;A01N43/78;A01N43/836;C07D405/06;C07D417/06;

  • 国家 AR

  • 入库时间 2022-08-21 14:27:37

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