首页> 外国专利> PROCESS FOR THE PREPARATION OF 1S- 1 alpha, 2-ALPHA, 3 beta (1S *, 2R *), 5 beta - 3- 7- 2- (3,4-difluorophenyl) -CYCLOPROPYLAMINO -5- (propylthio) -3 H -1,2,3-triazolo 4,5-d pyrimidin-3-yl -5- (2-hydroxyethoxy) cyclopentane-1,2-dIOL AND ITS INTERMEDIATES

PROCESS FOR THE PREPARATION OF 1S- 1 alpha, 2-ALPHA, 3 beta (1S *, 2R *), 5 beta - 3- 7- 2- (3,4-difluorophenyl) -CYCLOPROPYLAMINO -5- (propylthio) -3 H -1,2,3-triazolo 4,5-d pyrimidin-3-yl -5- (2-hydroxyethoxy) cyclopentane-1,2-dIOL AND ITS INTERMEDIATES

机译:制备[1S- [1α,2-α,3β(1S *,2R *),5β]的方法]-3- [7- [2-(3,4-二氟苯基)-环丙胺基]- 5-(丙硫基)-3 H -1,2,3-三唑[4,5-d]嘧啶-3-基] -5-(2-羟基乙氧基)环戊烷-1,2-dIOL及其中间体

摘要

The present invention is directed to a process for preparing [1S-[1 Alpha,2 Alpha,3 Beta(1S*,2R*),5 Beta]]- 3-[7-[2-(3,4-difluorophenyl)-cyclopropylamino]-5-(propylthio)-3H-1,2,3-triazolo[4,5- d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)cyclopentane-l,2-diol and to intermediates useful in the process.
机译:本发明涉及制备[1S- [1α,2α,3β(1S *,2R *),5β]]-3- [7- [2-(3,4-二氟苯基)的方法-环丙基氨基] -5-(丙硫基)-3H-1,2,3-三唑并[4,5-d]嘧啶-3-基] -5-(2-羟基乙氧基)环戊烷-1,2-二醇及中间体在此过程中很有用。

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