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PHOSPHATE OF EPIDERMAL GROWTH FACTOR RECEPTOR INHIBITOR, CRYSTALLINE FORM OF PHOSPHATE, AND PREPARATION METHOD

机译:表皮生长因子受体抑制剂的磷酸盐,磷酸盐的结晶形式及其制备方法

摘要

The present invention relates to a phosphate crystalline form A of the compound of formula (I), and a preparation method for the phosphate crystalline form A. The phosphate crystalline form A has advantageous properties such as good solubility, low hygroscopicity and process developability. The preparation method is simple and low-cost, and has significant value for the future optimisation and development of the drug.
机译:本发明涉及式(I)的化合物的磷酸盐结晶形式A,以及该磷酸盐结晶形式A的制备方法。该磷酸盐结晶形式A具有有利的性质,例如良好的溶解性,低吸湿性和工艺可开发性。该制备方法简单,成本低廉,对药物的未来优化和开发具有重要的价值。

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