首页> 外国专利> HEXAHYDRODIBENZOA,GQUINOLIZINE COMPOUND, MANUFACTURING METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF

HEXAHYDRODIBENZOA,GQUINOLIZINE COMPOUND, MANUFACTURING METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF

机译:六乙双苯并[A,G]喹诺嗪化合物,其制备方法,药物组合物及其应用

摘要

PROBLEM TO BE SOLVED: To provide a novel hexahydrodibenzo[a,g]quinolizine compound having strong effect for treating diseases such as neurological diseases related to a dopamine receptor and a serotonin receptor, especially Parkinson disease, schizophrenia, drug dependence and migraine.SOLUTION: There are provided a novel hexahydrodibenzo[a,g]quinolizine compound represented by the general formula (I) and a derivative thereof, enantiomers thereof, diastereomers, racemic bodies and a mixture thereof and a pharmaceutically acceptable salt thereof.SELECTED DRAWING: None
机译:解决的问题:提供一种新型的六氢二苯并[a,g]喹诺嗪化合物,该化合物具有强效的治疗能力,例如与多巴胺受体和5-羟色胺受体相关的神经系统疾病,尤其是帕金森病,精神分裂症,药物依赖性和偏头痛。提供了由通式(I)表示的新型六氢二苯并[a,g]喹啉嗪化合物及其衍生物,其对映异构体,非对映异构体,外消旋体及其混合物和药学上可接受的盐。

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