首页> 外国专利> N-ACETYLGLUCOSAMINE SUGAR CHAIN GROUP-CONTAINING COMPOUND, CARRIER COMPOUND FOR DRUG DELIVERY, DRUG PREPARATION, AND DRUG DELIVERY SYSTEM

N-ACETYLGLUCOSAMINE SUGAR CHAIN GROUP-CONTAINING COMPOUND, CARRIER COMPOUND FOR DRUG DELIVERY, DRUG PREPARATION, AND DRUG DELIVERY SYSTEM

机译:含N-乙酰氨基葡萄糖糖链组的化合物,用于药物输送,药物制备和药物输送系统的载体化合物

摘要

An N-acetylglucosamine sugar chain group-containing compound which can easily reach cells/sites on which a vimentin and/or desmin protein(s) is/are exposed, which compound has excellent affinity to N-acetylglucosamine sugar chain-recognizing proteins; a drug delivery carrier compound comprising the compound: a preparation using the drug delivery earner compound; and a drug delivery system; are provided. These are an N-acetylglucosamine sugar chain group-containing compound having a weight average molecular weight within the range of 15,000 to 100,000; a drug delivery carrier compound comprising the compound; a preparation using the drug delivery carrier compound; and a drug delivery system.
机译:含有N-乙酰氨基葡糖糖链基的化合物,可以容易地到达波形蛋白和/或结蛋白蛋白质暴露的细胞/部位,该化合物对识别N-乙酰氨基葡糖糖链的蛋白质具有优异的亲和力;药物递送载体化合物,其包含所述化合物:使用所述药物递送载体化合物的制剂;和药物输送系统;提供。它们是重均分子量为15,000〜100,000的含N-乙酰氨基葡糖糖链基的化合物。包含该化合物的药物递送载体化合物;使用药物递送载体化合物的制剂;和药物输送系统。

著录项

  • 公开/公告号US2017095564A1

    专利类型

  • 公开/公告日2017-04-06

    原文格式PDF

  • 申请/专利权人 SOMAR CORPORATION;

    申请/专利号US201515312507

  • 发明设计人 HIROHIKO ISE;

    申请日2015-05-19

  • 分类号A61B10;C08F12/26;A61K49;A61K41;

  • 国家 US

  • 入库时间 2022-08-21 13:46:24

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