首页> 外国专利> crystalline compound, pharmaceutical composition, use of crystalline compound, crystalline vortioxetine hydrobromide hydrate, method for preparation of crystalline vortioxetine hydrobromide hydrate, method for preparation of crystalline compound and use of crystalline vortioxetine hydrobromide hydrate

crystalline compound, pharmaceutical composition, use of crystalline compound, crystalline vortioxetine hydrobromide hydrate, method for preparation of crystalline vortioxetine hydrobromide hydrate, method for preparation of crystalline compound and use of crystalline vortioxetine hydrobromide hydrate

机译:结晶化合物,药物组合物,结晶化合物的用途,结晶伏立西汀氢溴酸盐水合物,结晶伏立西汀氢溴酸盐水合物的制备方法,结晶化合物的制备方法和结晶伏立西汀氢溴酸盐水合物的用途

摘要

abstract new crystalline form of vortioxetine hydrobromide The present invention relates to a crystalline compound comprising a hydrobromic acid (hbr) salt of a compound of formula i (1- {2 - [(2,4-dimethylphenyl) sulfanyl] phenyl} piperazine, inn: vortioxetine), with an xrpd pattern with characteristic peaks (expressed as 2 ± ± 0.2 ° 2 '(cuk? radiation)) at 5.5 °, 14.8 °, 16.7 ° and 20 ° , 0 °, and processes for obtaining the same. formula i
机译:氢伏替西汀的抽象新晶体形式本发明涉及一种结晶化合物,其包含式i化合物(1- {2-[((2,4-二甲基苯基)硫烷基]苯基}哌嗪的氢溴酸盐) :vortioxetine),其特征是在5.5°,14.8°,16.7°和20°,0°处具有特征峰(表示为2±±0.2°2'(cuk?辐射))的xrpd模式及其获得方法。公式一

著录项

  • 公开/公告号BR112015006075A2

    专利类型

  • 公开/公告日2017-07-04

    原文格式PDF

  • 申请/专利权人 SANDOZ AG;

    申请/专利号BR20151106075

  • 申请日2013-09-18

  • 分类号A61K31/495;A61P25;C07D295/096;

  • 国家 BR

  • 入库时间 2022-08-21 13:40:14

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