首页> 外国专利> ISOLATED INTERMEDIATE OF DAPAGLIFLOZIN, PROCESS FOR THE PREPARATION OF ISOLATED INTERMEDIATE OF DAPAGLIFLOZIN, PROCESS FOR THE PREPARATION OF DAPAGLIFLOZIN

ISOLATED INTERMEDIATE OF DAPAGLIFLOZIN, PROCESS FOR THE PREPARATION OF ISOLATED INTERMEDIATE OF DAPAGLIFLOZIN, PROCESS FOR THE PREPARATION OF DAPAGLIFLOZIN

机译:DAPAGLIFLOZIN的分离中间体,DAPAGLIFZIN的分离中间体的制备方法

摘要

Aspects of the present invention relates to an isolated intermediate of Dapagliflozin (Formula III) and its preparation, process for the preparation of Dapagliflozin, process for the preparation of crystalline propane-1,2,3-triol solvate of dapagliflozin, process for the preparation of L-proline complex of Dapagliflozin, solid premix of dapagliflozin with the polymer selected from the group consisting of eudragit, syloid, MCC Avicel PH 102 (1:1) and MCC Avicel PH 102 (1:2).
机译:本发明的方面涉及达格列净的分离的中间体(式III)及其制备,达格列净的制备方法,达格列净的结晶丙烷-1,2,3-三醇溶剂化物的制备方法,制备方法达格列净的L-脯氨酸复合物,达格列净与聚合物的固体预混合物,该聚合物选自eudragit,syloid,MCC Avicel PH 102(1:1)和MCC Avicel PH 102(1:2)。

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