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INJECTION CONTAINING CAMPTOTHECIN DERIVATIVE, AND INJECTION LIQUID, PREPARATION AND USE THEREOF

机译:含有喜树碱衍生物的注射剂及其注射液,制备方法和用途

摘要

An injection containing a camptothecin derivative, and preparation method and use thereof. The injection comprises a solid-state portion and liquid-state portion separately packaged. The solid-state portion is a lyophilized powder, and the liquid-state portion comprises a solubilizer and water for injection. The lyophilized powder comprises a camptothecin derivative or a pharmaceutically acceptable salt thereof. The camptothecin derivative has the following structure (I).
机译:含有喜树碱衍生物的注射剂及其制备方法和用途。该注射剂包括分开包装的固态部分和液态部分。固态部分是冻干粉末,而液态部分包括增溶剂和注射用水。冻干粉末包含喜树碱衍生物或其药学上可接受的盐。喜树碱衍生物具有以下结构(I)。

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