首页> 外国专利> VILDAGLIPTIN-CONTAINING PHARMACEUTICAL COMPOSITION, METHOD FOR STABILIZING VILDAGLIPTIN IN PHARMACEUTICAL COMPOSITION, AND STABILIZER OF VILDAGLIPTIN

VILDAGLIPTIN-CONTAINING PHARMACEUTICAL COMPOSITION, METHOD FOR STABILIZING VILDAGLIPTIN IN PHARMACEUTICAL COMPOSITION, AND STABILIZER OF VILDAGLIPTIN

机译:含维格列汀的药物组合物,在药物组合物中稳定维格列汀的方法和维他汀的稳定剂

摘要

PROBLEM TO BE SOLVED: To provide a vildagliptin-containing pharmaceutical composition capable of improving the influence of dispensing environment, preservation environment, etc., in particular, decrease in the stability of vildagliptin due to the influence of high humidity; a method for stabilizing vildagliptin in pharmaceutical composition; and a stabilizer of vildagliptin.;SOLUTION: According to the present invention, there is provided a vildagliptin-containing pharmaceutical composition comprising vildagliptin and at least one selected from the group consisting of mannitol, lactose, and corn starch. The total content of at least one member selected from the group consisting of mannitol, lactose, and corn starch is 50% by mass or more.;SELECTED DRAWING: None;COPYRIGHT: (C)2018,JPO&INPIT
机译:解决的问题:提供一种含维格列汀的药物组合物,其能够改善分配环境,保存环境等的影响,尤其是由于高湿度的影响而使维格列汀的稳定性降低;使药物组合物中的维格列汀稳定的方法;解决方案:根据本发明,提供了一种含维达列汀的药物组合物,其包含维达列汀和选自甘露醇,乳糖和玉米淀粉的至少一种。选自甘露醇,乳糖和玉米淀粉中的至少一种的总含量为50质量%以上。;选图:无;版权:(C)2018,JPO&INPIT

著录项

  • 公开/公告号JP2017222592A

    专利类型

  • 公开/公告日2017-12-21

    原文格式PDF

  • 申请/专利权人 ELMED EISAI KK;

    申请/专利号JP20160118230

  • 发明设计人 IKEDA HIROMI;

    申请日2016-06-14

  • 分类号A61K31/40;A61P3/10;A61K47/10;A61K47/26;A61K47/36;

  • 国家 JP

  • 入库时间 2022-08-21 13:10:39

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