首页> 外国专利> COMPOSITION AND METHODS TO IMPROVE STABILITY, DOSING, PHARMACODYNAMICS AND PRODUCT SHELF LIFE OF ENDOCANNABINOIDS, PHYTOCANNABINOIDS AND SYNTHETIC CANNABINOIDS DELIVERED BY NASAL INHAER

COMPOSITION AND METHODS TO IMPROVE STABILITY, DOSING, PHARMACODYNAMICS AND PRODUCT SHELF LIFE OF ENDOCANNABINOIDS, PHYTOCANNABINOIDS AND SYNTHETIC CANNABINOIDS DELIVERED BY NASAL INHAER

机译:改善鼻腔吸入器释放的内大麻素,植物大麻素和合成大麻素的稳定性,剂量,药动学和产品保质期的组合物和方法

摘要

An inhaler-delivery-device-packaged homogenate of solid heterogeneous-lipid particulates carrying lipophilic cannabinoid receptor agonists and/or antagonists, wherein the solid heterogeneous-lipid particles comprises: one (or more) lipid(s) whose melting point(s) is (are) substantially above room temperature; in combination with, one (or more) lipid(s) whose melting point(s) is (are) substantially less than room temperature.
机译:吸入递送装置包装的,带有亲脂性大麻素受体激动剂和/或拮抗剂的固体异质脂质颗粒的匀浆,其中所述固体异质脂质颗粒包含:(一种或多种)脂质,其熔点为显着高于室温;与一种或多种熔点实质上低于室温的脂质组合。

著录项

  • 公开/公告号US2018000727A1

    专利类型

  • 公开/公告日2018-01-04

    原文格式PDF

  • 申请/专利权人 MICHAEL WILLINSKY;

    申请/专利号US201615545500

  • 发明设计人 MICHAEL WILLINSKY;

    申请日2016-01-18

  • 分类号A61K9;A61K47/12;A61K31/352;A61K9/14;A61K9/12;A61K47/44;A61K36/18;

  • 国家 US

  • 入库时间 2022-08-21 13:00:39

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