首页> 外国专利> polymorphic solid or solvated form of 4- 2 - 5-methyl-1- (2-naphthalenyl) -1h-pyrazol-3-yl oxy ethyl morpholine hydrochloride salt, solid form, process for preparation polymorphic phase form i, polymorphic phase form iii, polymorphic phase form ii, polymorphic phase form iv, dioxane solvate, chloroform solvate, use of polymorphic phase form ii, polymorphic phase form iii, polymorphic phase form iv, dioxane solvate or chloroform solvate, process for preparing phase 4- form of 4- 2 - 5-methyl-1- (2-naphthalenyl) -1h hydrochloride salt -pyrazol-3-yl oxy ethyl morpholine and pharmaceutical composition

polymorphic solid or solvated form of 4- 2 - 5-methyl-1- (2-naphthalenyl) -1h-pyrazol-3-yl oxy ethyl morpholine hydrochloride salt, solid form, process for preparation polymorphic phase form i, polymorphic phase form iii, polymorphic phase form ii, polymorphic phase form iv, dioxane solvate, chloroform solvate, use of polymorphic phase form ii, polymorphic phase form iii, polymorphic phase form iv, dioxane solvate or chloroform solvate, process for preparing phase 4- form of 4- 2 - 5-methyl-1- (2-naphthalenyl) -1h hydrochloride salt -pyrazol-3-yl oxy ethyl morpholine and pharmaceutical composition

机译:[[4- [2-[[5-甲基-1-(2-萘基)-1h-吡唑-3-基]氧基]乙基]吗啉]盐酸盐的多晶型固体或溶剂化形式,固体形式,制备多晶相形式的方法i,多晶相形式iii,多晶相形式ii,多晶相形式iv,二恶烷溶剂化物,氯仿溶剂化物,使用多晶相形式ii,多晶相形式iii,多晶相形式iv,二恶烷溶剂化物或氯仿溶剂化物,制备方法4- [2-[[[5-甲基-1-(2-萘基)-1h]盐酸盐-吡唑-3-基]氧基]乙基]吗啉的4-形式和药物组合物

摘要

polymorphic solid or solvated form of 4- [2 - [[5-methyl-1- (2-naphthalenyl) -1h-pyrazol-3-yl] oxy] ethyl] morpholine hydrochloride salt, solid form, process for preparation polymorphic phase form i, polymorphic phase form iii, polymorphic phase form ii, polymorphic phase form iv, dioxane solvate, chloroform solvate, use of polymorphic phase form ii, polymorphic phase form iii, polymorphic phase form iv, dioxane solvate or chloroform solvate, process for the preparation of phase form I of 4- [2 - [[5-methyl-1- (2-naphthalenyl) -1h- hydrochloride salt pyrazol-3-yl] oxy] ethyl] morpholine and pharmaceutical composition The present invention relates to polymorphs and solvates of 4- [2 - [[5-methyl-1- (2-naphthalenyl) -1hpyrazol-2-one hydrochloride salt. 3-yl] oxy] ethyl] morpholine (p027), process for their preparation, and pharmaceutical compositions comprising them.
机译:[[4- [2-[[5-甲基-1-(2-萘基)-1h-吡唑-3-基]氧基]乙基]吗啉]盐酸盐的多晶型固体或溶剂化物形式,固体形式,制备多晶相形式的方法i,多晶相形式iii,多晶相形式ii,多晶相形式iv,二恶烷溶剂化物,氯仿溶剂化物,使用多晶相形式ii,多晶相形式iii,多晶相形式iv,二恶烷溶剂化物或氯仿溶剂化物,制备方法4- [2-[[[5-甲基-1-(2-萘基)-1h-盐酸盐吡唑-3-基]氧基]乙基]吗啉的相形式I的制备和药物组合物本发明涉及多晶型物和溶剂化物4- [2-[[5-甲基-1-(2-萘基)-1]吡唑-2-盐酸盐。 3-基]氧基]乙基]吗啉(p027),其制备方法和包含它们的药物组合物。

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