SITE-SELECTIVE PEPTIDES AND PROTEIN LABELLING AND SYNTHESIS OF HOMOGENOUS PROTEIN CONJUGATES

摘要

The invention pertains to the method for the site selective modification of peptides and proteins comprising of the activation of the single site (Nɛ-NH2) of peptides and proteins and the method comprising one of formylation; interception of formylation; alkynylation or amino phosphonation of peptides and proteins.