首页> 外国专利> PHARMACEUTICAL COMBINATION OF ETHINYLESTRADIOL AND DROSPIRENONE FOR USE AS A CONTRACEPTIVE

PHARMACEUTICAL COMBINATION OF ETHINYLESTRADIOL AND DROSPIRENONE FOR USE AS A CONTRACEPTIVE

机译:乙炔雌二醇和屈螺酮的药物组合用作避孕药

摘要

A Pharmaceutical composition comprising, as a First Active Agent, 6beta, pharmacy, 15beta, 16beta - dimetilen - 3 - oxo - pregn 17alfa - - 4 - - 21- carbolactona (17 cases) in an amount corresponding to a Daily Dose to be administered with lacompo sicyon, from approximately 2mg approximately 4 mgAnd as a Second ACTIVE AGENT, 17alfa - ethinyl estradiol (estradiol) in an amount corresponding to a daily dose of from about 0.01 mgaproximadamente 0.05 mg,Jointly with one or more pharmaceutically acceptable carriers or excipients.In a specific implementation, a number of composicionconsiste Daily dosage units placed in a Packaging Unit, yseparables individually packaged separately,Yproporcionadas for oral Administration for a period of at least 21 consecutive days of daily dosing units, including the combining of drospirenone and ethinyl estradiol.The composition also puedecomprender 7 or less Daily dosage units containing no assets or agents that contain ethinyl estradiol.
机译:一种药物组合物,其包含作为第一活性剂的6beta,药房,15beta,16beta-dimetilen-3-oxo-pregn 17alfa--4-21- carbolactona(17例),其用量相当于每日给药的剂量Lacompo sicyon约2mg约4 mg,第二种活性剂17alfa-乙炔雌二醇(estradiol)的量相当于每日约0.01 mgaproximadamente 0.05 mg,并与一种或多种药学上可接受的载体或赋形剂一起使用。在一个具体的实施方案中,许多composicion由组成包装单位的每日剂量单位,单独包装的可分离物,用于口服的Yproporcionadas连续至少21天的每日剂量单位,包括屈螺酮和乙炔基雌二醇的组合。该组合物还可以不包含7个或更少的日剂量单位,不包含资产或含有乙炔雌二醇的药剂。

著录项

  • 公开/公告号RS50262B2

    专利类型

  • 公开/公告日2018-10-31

    原文格式PDF

  • 申请/专利权人 BAYER PHARMA AKTIENGESELLSCHAFT;

    申请/专利号RSP20020145

  • 申请日2000-08-31

  • 分类号A61K9/14;A61K31/565;A61K;A61K9/20;A61K9/28;A61K31/567;A61K31/569;A61K31/57;A61K31/58;A61K31/585;A61P;A61P5/28;A61P15;A61P15/18;

  • 国家 RS

  • 入库时间 2022-08-21 12:50:08

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