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COMPOUND FOR ACTIVATING ADENOSINE MONOPHOSPHATE-ACTIVATED PROTEIN KINASE

机译:激活腺苷单磷酸激活的蛋白激酶的化合物

摘要

Disclosed is a compound as represented by formula I. The compound is used as an activator for adenosine monophosphate-activated protein kinase to phosphorylate and activate adenosine monophosphate-activated protein kinase, and then to regulate a downstream signaling pathway, and thus can inhibit the growth and division of liver cancer cells and breast cancer cells, and can also induce the death of fat cells. Thus, the compound in the present invention can be applied in manufacturing of pharmaceutical compositions for adenosine monophosphate-activated protein kinase-related cancers and fat metabolism diseases or syndromes, and can also be used for treating adenosine monophosphate-activated protein kinase-related cancers and fat metabolism diseases or syndromes.
机译:公开了由式I表示的化合物。该化合物用作单磷酸腺苷活化的蛋白激酶的活化剂,以磷酸化和活化单磷酸腺苷活化的蛋白激酶,然后调节下游信号传导途径,因此可以抑制其生长。以及肝癌细胞和乳腺癌细胞的分裂,还可以诱导脂肪细胞死亡。因此,本发明的化合物可用于制造腺苷单磷酸激活的蛋白激酶相关的癌症和脂肪代谢疾病或综合征的药物组合物,还可用于治疗腺苷单磷酸激活的蛋白激酶相关的癌症和脂肪代谢疾病或综合症。

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