首页> 外国专利> SYNTHETIC METHOD OF FUSED HETEROAROMATIC COMPOUND AND FUSED HETEROAROMATIC COMPOUND AND INTERMEDIATE THEREFOR AND SYNTHETIC METHOD OF INTERMEDIATE

SYNTHETIC METHOD OF FUSED HETEROAROMATIC COMPOUND AND FUSED HETEROAROMATIC COMPOUND AND INTERMEDIATE THEREFOR AND SYNTHETIC METHOD OF INTERMEDIATE

机译:熔融杂铜化合物和熔融杂铜化合物及其中间体的合成方法和中间体的合成方法

摘要

The present invention relates to a synthesis method of a fused heteroaromatic compound, which comprises the steps of: reacting a compound represented by chemical formula 1 with a metal alkyl chalcogenide in the presence of a palladium catalyst and a tertiary phosphine catalyst to obtain a first intermediate represented by chemical formula 2; obtaining a second intermediate represented by chemical formula 3 from the first intermediate; obtaining a third intermediate from the second intermediate and a compound represented by chemical formula 4; obtaining a fourth intermediate including a chalcogen-containing ring from the third intermediate; and performing a cyclization reaction of the fourth intermediate to obtain a fused heteroaromatic compound. In addition, the present invention relates to a fused heteroaromatic compound obtained by the synthesis method, an intermediate thereof, and a synthesis method of the intermediate.
机译:本发明涉及一种稠合杂芳族化合物的合成方法,该方法包括以下步骤:在钯催化剂和叔膦催化剂的存在下,使化学式1表示的化合物与金属硫属金属化物反应,得到第一中间体。由化学式2表示;从第一中间体获得化学式3表示的第二中间体;由第二中间体和化学式4表示的化合物获得第三中间体;从第三中间体获得包括含硫属元素环的第四中间体;进行第四中间体的环化反应,得到稠合的杂芳族化合物。另外,本发明涉及通过合成方法获得的稠合杂芳族化合物,其中间体以及该中间体的合成方法。

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