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HETEROCYCLES AND THEIR RADIOLABELED ANALOGS USEFUL AS COX-1 SELECTIVE INHIBITORS

机译:杂环化合物及其放射标记的类似物可用作COX-1选择性抑制剂

摘要

The present invention relates to novel heterocycles which are potent and selective inhibitors of cyclooxygenase-1 (COX-1) and to their radiolabeled derivatives thereof which are both useful as theranostics of a number of pathologies.
机译:本发明涉及新型的杂环化合物,它们是有效的和选择性的环氧合酶-1(COX-1)抑制剂,并涉及其放射性标记的衍生物,它们均可用作多种病理学的治疗方法。

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