diespiro 1,2,4-trioxolane, pharmaceutical formulation, process for the preparation of a diespiro 1,2,4-trioxolane derivative, intermediate, and method for preventing and / or treating malaria and schistosomiasis or a cancer.

摘要

The present invention relates to novel trioxolane derivatives in the manufacture of a medicament for preventing or treating malaria. Specifically, the present invention relates to trioxolane derivatives useful for the preparation of a pharmaceutical formulation for inhibiting the proliferation of malaria parasites.