首页> 外国专利> ACTIVE METABOLITE OF 1 - (2-BROMPHENYL) SULPHONYL -5-METHOXY-3 - (4-METHYL-1-PIPERAZINYL) METHYL -1H-INDOL-DIMESYLATE-MONOHYDRATE AND DIMESYLATE-DIHYDRATE SALT

ACTIVE METABOLITE OF 1 - (2-BROMPHENYL) SULPHONYL -5-METHOXY-3 - (4-METHYL-1-PIPERAZINYL) METHYL -1H-INDOL-DIMESYLATE-MONOHYDRATE AND DIMESYLATE-DIHYDRATE SALT

机译:1-[((2-溴苯甲基)磺酰基] -5-甲氧基-3-[(4-甲基-1-哌嗪基)甲基] -1H-吲哚-二甲苯磺酸一铵和二甲苯磺酸二甲酯盐的活性代谢产物

摘要

The present invention is directed to active metabolite of 1-[(2-bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole dimesylate monohydrate of formula (I). The present invention is also directed to dimesylate dihydrate salt of formula (II). The compounds of formula (I) and formula (II) are useful in the treatment of various disorders that are related to 5-HT6 receptor antagonist.
机译:本发明涉及式(I)的1-[(2-溴苯基)磺酰基] -5-甲氧基-3-[(4-甲基-1-哌嗪基)甲基] -1H-吲哚二甲酸酯一水合物的活性代谢物。本发明还涉及式(II)的二甲磺酸二水合物盐。式(I)和式(II)的化合物可用于治疗与5-HT 6受体拮抗剂有关的各种疾病。

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