首页> 外国专利> INTERMEDIATE FOR SYNTHESIS OF 1-(2-DEOXY-2-FLUORO-4-THIO-beta-D-ARABINOFURANOSYL) CYTOSINE, INTERMEDIATE FOR SYNTHESIS OF THIONUCLEOSIDE, AND METHODS FOR PRODUCING THESE INTERMEDIATES

INTERMEDIATE FOR SYNTHESIS OF 1-(2-DEOXY-2-FLUORO-4-THIO-beta-D-ARABINOFURANOSYL) CYTOSINE, INTERMEDIATE FOR SYNTHESIS OF THIONUCLEOSIDE, AND METHODS FOR PRODUCING THESE INTERMEDIATES

机译:合成1-(2-脱氧-2-氟-2-氟-β-D-阿拉伯呋喃核糖基)胞嘧啶的中间体,合成硫核苷的中间体以及制备这些中间体的方法

摘要

A compound represented by a formula [ID] as shown below (wherein R 1A , R 1B , R 2A , R 2B , R 3A and R 3B represent a hydrogen atom, an optionally substituted C 1-6 alkyl group, and the like) is useful as an intermediate for producing a thionucleoside, and the production method of the present invention is useful as a method for producing a thionucleoside.
机译:如下所示的由式[ID]表示的化合物(其中R 1A,R 1B,R 2A,R 2B,R 3A和R 3B表示氢原子,任选取代的C 1-6烷基等)本发明的制备方法可用作制备硫代核苷的中间体,本发明的制备方法可用作制备硫代核苷的中间体。

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