首页> 外国专利> COMPOSITION FOR EVALUATING ACTIVITY OF DRUG METABOLIZING ENZYME OF NEW DRUG CANDIDATE, AND METHOD FOR EVALUATING ACTIVITY OF DRUG METABOLIZING ENZYME BY USING SAME

COMPOSITION FOR EVALUATING ACTIVITY OF DRUG METABOLIZING ENZYME OF NEW DRUG CANDIDATE, AND METHOD FOR EVALUATING ACTIVITY OF DRUG METABOLIZING ENZYME BY USING SAME

机译:药物新药候选药物评估药物代谢酶活性的组成以及药物代谢酶活性评估的方法

摘要

The present invention relates to a composition containing a cocktail set for evaluating the activity of a drug metabolizing enzyme of a novel drug candidate, and a method for evaluating the activity of a drug metabolizing enzyme of a novel drug candidate by using the same. When the composition and the method are used, the activity of 10 types of cytochrome P450 isozymes can be simultaneously evaluated such that effects on the activity of a drug metabolizing enzyme of a novel drug candidate can be rapidly measured, thereby enabling drug interactions in the body to be predicted.
机译:本发明涉及一种包含用于评价新型候选药物的药物代谢酶活性的鸡尾酒组合物的组合物,以及通过使用该组合物评价新型候选药物的药物代谢酶活性的方法。当使用该组合物和方法时,可以同时评估10种细胞色素P450同工酶的活性,从而可以快速测量对新型候选药物的药物代谢酶活性的影响,从而使体内的药物相互作用成为可能。待预测。

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