COMPOSITIONS FOR INHIBITION OF THE METHYLTRANSFERASE SETD6

摘要

Described herein are synthetic polypeptide inhibitors of the SET-domain-containing protein 6 (SETD6) methyltransferase, and polypeptide chimeras thereof including at least one cell penetrating peptide. Pharmaceutical compositions and uses thereof for treatment of diseases and conditions associated with overexpression of SETD6 are also described.