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COX-2-TARGETING, PLATINUM-CONTAINING CONJUGATES AND THEIR USE IN THE TREATMENT OF TUMORS AND CANCERS
COX-2-TARGETING, PLATINUM-CONTAINING CONJUGATES AND THEIR USE IN THE TREATMENT OF TUMORS AND CANCERS
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机译:COX-2靶向,含铂结合物及其在肿瘤和癌症治疗中的用途
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摘要
The present disclosure provides platinum-containing conjugates that selectively target and kill tumor/cancer cells. The conjugates contain a moiety that selectively targets COX-2, which is overexpressed by a broad range of tumor/cancer cells..
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机译:本公开提供了选择性靶向并杀死肿瘤/癌细胞的含铂缀合物。缀合物包含选择性靶向COX-2的部分,该部分被多种肿瘤/癌细胞过度表达。 <图像文件=“ IMGA0001.GIF” he =“ 30” imgContent =“ chem” imgFormat =“ GIF” wi =“ 136” /> Chemistry> <化学id =“ chema02” > <图像文件=“ IMGA0002.GIF” he =“ 30” imgContent =“ chem” imgFormat =“ GIF” wi =“ 138” /> Chemistry> <图像文件=“ IMGA0003 .GIF“ he =” 27“ imgContent =” chem“ imgFormat =” GIF“ wi =” 149“ /> Chemistry> <图像文件=” IMGA0004.GIF“ he =” 35 “ imgContent =” chem“ imgFormat =” GIF“ wi =” 80“ /> Chemistry>。
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