COMPOUND, PHARMACEUTICAL COMPOSITION, USE OF A COMPOUND, PROCESS FOR THE PREPARATION OF A COMPOUND, NEW INTERMEDIATE AND PROCESS FOR THE PREPARATION OF A NEW INTERMEDIATE

摘要

"compound, pharmaceutical composition, use of a compound, method for treatment, method for reducing the morbidity and mortality associated with being overweight, process for the preparation of a compound, new intermediate and process for the preparation of a new intermediate ". the present invention relates to tetracyclic indoles of arylsulfonyl, their derivatives, their analogues, their tautomeric forms, their stereo isomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates, the innovative intermediates described herein and the pharmaceutically acceptable compositions containing the same. the present invention is particularly related to new tetracyclic indoles of arylsulfonyl having the general formula (i), its derivatives, its analogs, tautomeric forms, its stereo isomers, its polymorphs, its pharmaceutically acceptable salts, its pharmaceutically acceptable solvates, to the innovative intermediates here described and the pharmaceutically acceptable compositions containing them. the present invention also relates to the process (es) for the preparation of such compound (s) having the general formula (i), to compositions containing effective amount (s) of said compound and to the use of such a compound / composition in therapies.