首页> 外国专利> -5-35---1--3--4-4---1--2---4-- PROCESS FOR THE PREPARATION OF N-5-35-DIFLUORO-BENZYL-1H-INDAZOL-3-YL-4-4-METHYL-PIPERAZIN-1-YL-2-TETRAHYDRO-PYRAN-4-YLAMINO-BENZAMIDE

-5-35---1--3--4-4---1--2---4-- PROCESS FOR THE PREPARATION OF N-5-35-DIFLUORO-BENZYL-1H-INDAZOL-3-YL-4-4-METHYL-PIPERAZIN-1-YL-2-TETRAHYDRO-PYRAN-4-YLAMINO-BENZAMIDE

机译:-[5-35 --- 1--3-]-4-4 --- 1--2 --- 4-- N- [5-35-DIFLUORO-BENZYL-1H-吲唑的制备方法-3-YL] -4-4-甲基哌嗪-1-基-2-四氢吡喃-4-基氨基苯甲酰胺

摘要

The present invention is N-[5-(3,5-difluoro-benzyl)-1H-indazol-3-yl]-4-(4-methyl-piperazin-1-yl)-2-(tetrahydro It relates to a method for preparing -pyran-4-ylamino)-benzamide. Novel solid forms of the compounds, the utility of these solid forms in treating diseases caused by unregulated protein kinase activity, and pharmaceutical compositions containing them are also objects of the present invention.
机译:N- [5-(3,5-二氟苄基)-1H-吲唑-3-基] -4-(4-甲基哌嗪-1-基)-2-(四氢) -吡喃-4-基氨基)-苯甲酰胺的制备方法。化合物的新型固体形式,这些固体形式在治疗由不受调节的蛋白激酶活性引起的疾病中的用途以及包含它们的药物组合物也是本发明的目的。

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