机译:发现4,5,6,7-四氢苯并1,2-d噻唑作为靶向ATP结合位点的新型DNA旋转酶抑制剂
Univ Ljubljana, Fac Pharm, Ljubljana 1000, Slovenia;
Natl Inst Chem, Lab Biocomp & Bioinformat, Ljubljana 1001, Slovenia;
Univ Helsinki, Fac Pharm, Ctr Drug Res, FI-00014 Helsinki, FinlandGalapagos Istrazivacki Ctr Doo, HR-10000 Zagreb, Croatia;
机译:Computer-aided structure-based optimization of 4,5,6,7-tetrahydrobenzodthiazole-2,6-diamine derivatives as DNA gyrase B inhibitors
机译:ChemInform Abstract: Convenient Heterocyclization Reactions with Ethyl 2‐Amino‐4,5,6,7‐ tetrahydrobenzo(b)thiophene‐3‐carboxylate: Synthesis of Thiazole, Isoxazole, Pyrazole, Pyrimidine and Pyridazine Derivatives.
机译:Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold- Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa