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机译:苯基吡唑并1,5-a喹唑啉-5(4 H)-酮:用于开发非喜树碱拓扑异构酶 i (Top1) 抑制剂的合适支架
Department of Pharmacy, University of Naples Federico II, Via D. Montesano 49, 80131 Napoli, Italy;
Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, Bethesda, MD 20892-4255, United States;
Istituto Pasteur - Fondazione Cenci Bolognetti, Dipartimento di Chimica e Tecnologie Del Farmaco, Sapienza Università di Roma, P.le Aldo Moro 5, I-00185, Rome, ItalyDepartment of Pharmacy, University of Pisa, via Bonanno 6, 56126 Pisa, ItalyDepartment of Drug Discovery and Development, Istituto Italiano di Tecnologia (IIT), Via Morego 30, 16163 Genova, ItalyDiSTABiF, Seconda Università di Napoli, Via G. Vivaldi 43, 81100 Caserta, Italy;
Phenylpyrazolo1; 5-aquinazolin-5(4 H)-one; suitable scaffold; noncamptothecin topoisomerase;
机译:Lamellarin-inspired potent topoisomerase I inhibitors with the unprecedented benzog1benzopyrano4,3-bindol-6(13H)-one scaffold
机译:Design, synthesis and biological evaluation of lapachol derivatives possessing indole scaffolds as topoisomerase I inhibitors
机译:Fragment-Based Drug Design, 2D-QSAR and DFT Calculation: Scaffolds of 1, 2, 4, triazolo 1, 5-a pyrimidin-7-amines as Potential Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase