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机译:Discovery of trypanocidal coumarins with dual inhibition of both the glycerol kinase and alternative oxidase of Trypanosoma brucei brucei
Ahmadu Bello Univ, Dept Biochem, Zaria 2222, Nigeria;
Univ Tokyo, Dept Biomed Chem, Grad Sch Med, Tokyo, Japan;
Kyoto Inst Technol, Grad Sch Sci & Technol, Dept Appl Biol, Kyoto, JapanUniv Sussex, Biochem & Med, Sch Life Sci, Brighton, E Sussex, EnglandRIKEN, Syst & Struct Biol Ctr, Yokohama, Kanagawa, JapanJuntendo Univ, Sch Med, Dept Mol & Cellular Parasitol, Tokyo, JapanUniv Tokyo, Grad Sch Pharmaceut Sci, Tokyo, JapanUniv Edinburgh, Ctr Immun Infect & Evolut, Edinburgh, Midlothian, Scotland;
energy metabolism; African trypanosomiasis; rational drug design; inhibitor; screening;