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机译:Discovery of a Novel Series of Orally Bioavailable and CNS Penetrant Glucagon-like Peptide-1 Receptor (GLP-1R) Noncompetitive Antagonists Based on a 1,3-Disubstituted-7-aryl-5,5-bis(trifluoromethyl)-5,8-dihydropyrimido4,5-dpyrimidine-2,4(1H,3H)-dione Core
Vanderbilt Univ, Sch Med, Vanderbilt Inst Chem Biol, Nashville, TN 37232 USA;
Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37232 USA;
Vanderbilt Univ, Sch Med, Vanderbilt Diabet Ctr, Nashville, TN 37232 USAVanderbilt Univ, Sch Med, Dept Med, Div Diabet Endocrinol & Metab, Nashville, TN 37232 USAVanderbilt Univ, Sch Med, Vanderbilt Ctr Neurosci Drug Discovery, Nashville, TN 37232 USA;