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机译:13C和1H-NMR研究丝氨酸蛋白酶对氧和四面体中间稳定的研究:通过研究肽衍生的氯甲烷和G对丝氨酸蛋白酶抑制的抑制剂特异性和效力,优化抑制剂弹头特异性和效力
UCD School of Biomolecular and Biomedical Science, Centre for Synthesis and Chemical Biology, UCD Conway Institute, University College Dublin, Dublin 4, Ireland. J.Paul.G.Malthouse@ucd.ie;
Serine Endopeptidases; warhead; glyoxalSerine ProteinaseOXOANIONMethyl Chloride1H NMRPotency;