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机译:蛋白质精氨酸甲基转移酶6的第一类,高度选择性和细胞活性的变构抑制剂6
Icahn Sch Med Mt Sinai Mt Sinai Ctr Therapeut Discovery Tisch Canc Inst Dept Pharmacol Sci New York NY 10029 USA;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Icahn Sch Med Mt Sinai Mt Sinai Ctr Therapeut Discovery Tisch Canc Inst Dept Pharmacol Sci New York NY 10029 USA;
Icahn Sch Med Mt Sinai Mt Sinai Ctr Therapeut Discovery Tisch Canc Inst Dept Pharmacol Sci New York NY 10029 USA;
Icahn Sch Med Mt Sinai Mt Sinai Ctr Therapeut Discovery Tisch Canc Inst Dept Pharmacol Sci New York NY 10029 USA;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Ontario Inst Canc Res Toronto ON M5G 0A3 Canada;
Ontario Inst Canc Res Toronto ON M5G 0A3 Canada;
Eli Lilly &
Co Lilly Res Labs Indianapolis IN 46225 USA;
Eli Lilly &
Co Lilly Res Labs Indianapolis IN 46225 USA;
Eli Lilly &
Co Lilly Res Labs Indianapolis IN 46225 USA;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Ontario Inst Canc Res Toronto ON M5G 0A3 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Icahn Sch Med Mt Sinai Mt Sinai Ctr Therapeut Discovery Tisch Canc Inst Dept Pharmacol Sci New York NY 10029 USA;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Univ Toronto Struct Genom Consortium Toronto ON M5G 1L7 Canada;
Icahn Sch Med Mt Sinai Mt Sinai Ctr Therapeut Discovery Tisch Canc Inst Dept Pharmacol Sci New York NY 10029 USA;
机译:精氨酸甲基转移酶3(PRMT3)的有效,选择性和细胞活性变构抑制剂。
机译:蛋白质精氨酸甲基转移酶4和蛋白质精氨酸甲基转移酶6的有效,选择性和细胞活性双重抑制剂的发现。
机译:人类I型精氨酸甲基转移酶的有效,选择性和细胞活性抑制剂。
机译:组合化学和亲和力色谱法系统探测蛋白 - 配体相互作用:应用于人甜菜碱的高选择性抑制剂的应用:同型半胱氨酸S-甲基转移酶
机译:用表面等离子体共振(SPR)靶向蛋白质精氨酸甲基转移酶-5(PRMT5)的小分子抑制剂的动力学分析
机译:精氨酸甲基转移酶3(PRMT3)的有效选择性和细胞活性变构抑制剂。
机译:发现有效,选择性和细胞活性双抑制剂的蛋白质精氨酸甲基转移酶4和蛋白质精氨酸甲基转移酶6
机译:哺乳动物组织中的胰蛋白酶样酶:取代异香豆素机制为基础的抑制剂,苯甲脒衍生物的底物特异性和Inhibitorypotency和精氨酸氟烷酮过渡态抑制剂