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机译:一种简单且无标记的电化学方法,用于检测β位淀粉样蛋白前体蛋白裂解酶并筛选其抑制剂
College of Chemistry and Chemical Engineering, Anyang Normal University, Anyang, Henan 455000, People's Republic of China;
College of Chemistry and Chemical Engineering, Anyang Normal University, Anyang, Henan 455000, People's Republic of China;
College of Chemistry and Chemical Engineering, Anyang Normal University, Anyang, Henan 455000, People's Republic of China;
College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu, Henan 476000, People's Republic of China;
College of Chemistry and Chemical Engineering, Anyang Normal University, Anyang, Henan 455000, People's Republic of China,College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu, Henan 476000, People's Republic of China;
Alzheimer's disease; Beta-amyloid; BACE1 inhibitor; Electrocatalysis; Heme;
机译:HIV蛋白酶抑制剂通过β位淀粉样蛋白前体蛋白切割酶-1平移上调改变淀粉样蛋白前体蛋白质处理
机译:从片段筛选到体内功效:优化一系列2-氨基喹啉作为β位淀粉样蛋白前体蛋白裂解酶1(bace1)的有效抑制剂
机译:P-糖蛋白外排和其他因素限制了小鼠中β-位淀粉样蛋白前体蛋白裂解酶1抑制剂对脑淀粉样蛋白的还原作用。
机译:基于Pharmacophore的虚拟筛选,分子对接和密度泛函理论方法,以发现有效的β-淀粉样蛋白前体蛋白(B-APP)抑制剂
机译:β-内啡肽抑制表达高水平突变淀粉样蛋白前体蛋白的SK-N-SH神经母细胞瘤细胞中淀粉样蛋白前体蛋白的表达。
机译:Beta站点淀粉样蛋白前体蛋白裂解酶1(BACE1)介导的野生型和转基因小鼠体内内源性淀粉样β的变化
机译:通过阻碍淀粉样蛋白途径(V0.1),“乙酰立位蛋白裂解酶-1的β-位点蛋黄酱切割酶-1的β-位点乳糖裂解酶-1的抑制剂,抑制APP-PS1-HEK293细胞中的分泌抑制蛋白前体蛋白的分泌”