Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G

Eugen Merkul; Elisabeth Schaefe; Thomas J. J. Mueller

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Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G

机译：一锅增田硼化-铃木偶联序列快速合成双（杂）芳基及其在简化子午线A和G的总合成中的应用

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3-(Hetero)aryl substituted indoles, 7-azaindoles, and pyrroles can be obtained in a very concise fashion via a one-pot Masuda borylation-Suzuki coupling sequence. The concise total syntheses of the marine natural products meridianins A (5) and G (4i) nicely illustrate the utility of this methodology.

机译：经由一锅增田（Masuda）硼酸酯化-铃木（Suzuki）偶联序列可以非常简洁的方式获得3-（杂）芳基取代的吲哚，7-氮杂吲哚和吡咯。海洋天然产物子午线虫A（5）和G（4i）的简洁的整体合成很好地说明了该方法的实用性。

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《Organic & biomolecular chemistry》 |2011年第9期|p.3139-3141|共3页
作者
Eugen Merkul; Elisabeth Schaefe; Thomas J. J. Mueller;
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Lehrstuhl fur Organische Chemie, Institut fuer Organische Chemie und Makromolekulare Chemie, Heinrich-Heine- Universitat Diisseldorf, Universitdtsstrasse 1, D-40225, Duesseldorf, Germany;

Lehrstuhl fur Organische Chemie, Institut fuer Organische Chemie und Makromolekulare Chemie, Heinrich-Heine- Universitat Diisseldorf, Universitdtsstrasse 1, D-40225, Duesseldorf, Germany;

Lehrstuhl fur Organische Chemie, Institut fuer Organische Chemie und Makromolekulare Chemie, Heinrich-Heine- Universitat Diisseldorf, Universitdtsstrasse 1, D-40225, Duesseldorf, Germany;

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Rapid synthesis of bis(hetero)aryls by one-pot Masuda borylation-Suzuki coupling sequence and its application to concise total syntheses of meridianins A and G

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