A gold (III) complex, a conjugate of a gold (III) complex, a pharmaceutical composition comprising a gold (III) complex, a method of producing a gold (III) complex and its use.

摘要

Problem to be solved: to provide a pharmaceutical composition containing a gold (III) complex and a method for producing the same.The gold (III) complex of the present invention has the following chemical formula (I).R1From aryl and amineR2From the first group (alkyl and cycloalkyl)R3HydrogenHalogenNitroCyanoAlkylAlkaline oxiAlkyl aminoAmino dialkylHydroxyalkylTrialkylsilylAryl dialkylsilylAlkaline TrioCycloalkylGroup 2HeterocyclePolycyclicAmino acidsPeptideFrom carbohydrate derivativesR4The first groupAlkyl alkoxyAlkyl aminoDialkyl aminoAlkaline TrioTrialkylphosphinoDialkylaryl phosphinoAlkyl diarylphosphinoTriarylphosphinoFrom the second groupIndependently selected.