首页> 外国专利> COMPOSITIONS IN THE FORM OF AN INJECTABLE AQUEOUS SOLUTION COMPRISING AMYLIN, AN AMYLIN RECEPTOR AGONIST OR AN AMYLIN ANALOG, AT LEAST ONE IONIC SPECIES AND AN AMPHIPHILIC COMPOUND CONTAINING HYDROPHOBIC RADICALS

COMPOSITIONS IN THE FORM OF AN INJECTABLE AQUEOUS SOLUTION COMPRISING AMYLIN, AN AMYLIN RECEPTOR AGONIST OR AN AMYLIN ANALOG, AT LEAST ONE IONIC SPECIES AND AN AMPHIPHILIC COMPOUND CONTAINING HYDROPHOBIC RADICALS

机译:包含淀粉蛋白,淀粉受体激动剂或淀粉蛋白类似物,至少一种含有疏水性自由基的两亲物质的组合物的组合物

摘要

The invention relates to a composition in the form of an injectable solution, comprising: amylin, an amylin receptor agonist or an amylin analog; at least one ionic species; and an amphiphilic compound comprising a hydrophilic skeleton HB, substituted by at least one hydrophobic radical -Hy of formula (I). The invention further relates to a composition according to the invention, characterised in that it also comprises prandial insulin. In one embodiment, the composition also comprises GLP- 1, GLP-1 analogs, and GLP-1 receptor agonists, commonly called GLP-1 RA.
机译:本发明涉及一种可注射溶液形式的组合物,包括:淀粉蛋白,淀粉蛋白受体激动剂或淀粉蛋白类似物;至少一种离子物种;和包含亲水性骨架Hb的两亲性化合物,被至少一种式(I)的疏水基团-Hy取代。本发明还涉及根据本发明的组合物,其特征在于它还包括伪装胰岛素。在一个实施方案中,该组合物还包括GLP-1,GLP-1类似物和GLP-1受体激动剂,通常称为GLP-1Ra。

著录项

  • 公开/公告号EP3829624A1

    专利类型

  • 公开/公告日2021-06-09

    原文格式PDF

  • 申请/专利权人 ADOCIA;

    申请/专利号EP20190752454

  • 发明设计人 DAUTY EMMANUEL;

    申请日2019-08-03

  • 分类号A61K38/22;A61K38/28;A61K45/06;A61K47/30;A61P3/10;

  • 国家 EP

  • 入库时间 2022-08-24 19:16:14

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