An estrogen sulfotransferase inhibitor composition comprises a compound of the formula ##STR1## wherein R.sub.1 is F, Br, NO.sub.2, or H; R.sub.2 is F, Br, NO.sub.2, NH.sub.2, or H; R is H or alkyl of 1-4 carbon atoms; R.sub.3 is O or H.sub.2 ; and R.sub.4 is H.sub.2, O, or . alpha.-H, &bgr;-OH; R.sub.5 is H.sub.2, &agr;-H and &bgr;-OH or B-H and &agr;-OH in admixture with a pharmaceutically acceptable carrier with the proviso that R.sub.1, R.sub.2 and R.sub.3 cannot all be hydrogen and one of R.sub.1 and R.sub.2 is F.
展开▼
机译：雌激素磺基转移酶抑制剂组合物包含式## STR1 ##的化合物，其中R 1是F，Br，NO 2或H; R 2是F，Br，NO 2，NH 2或H; R为H或1-4个碳原子的烷基; R.sub.3是O或H.sub.2; R.sub.4是H.sub.2，O或。 α.-H，＆bgr; -OH; R.sub.5是H.sub.2，α-H和b-OH或BH和α-OH与可药用载体混合，条件是R.sub.2 R 3不能全部是氢，R 1和R 2之一是F。
展开▼
