首页> 外国专利> nya derivat av bicykliska aminosyror, foerfarande foer deras framstaellning, year innehaollande medel och deras anvaendning.

nya derivat av bicykliska aminosyror, foerfarande foer deras framstaellning, year innehaollande medel och deras anvaendning.

机译:双环氨基酸的新衍生物,其制备方法,所含物质的年限及其用途。

摘要

The derivatives have the formula I …IMAGE… in which n is 0, 1 or 2, R is hydrogen, alkyl or aralkyl, R1 is hydrogen or alkyl, alkenyl, cycloalkyl, cycloalkenyl, cycloalkylalkyl, optionally substituted aryl or partially hydrogenated aryl, aryl-(C1-C4)-alkyl or aroyl-C1-alkyl, both of which can be substituted, a mono- or bicyclic heterocyclic radical or a side chain of a naturally occurring amino acid, R2 is hydrogen, alkyl, alkenyl or aralkyl, X is alkyl, alkenyl, cycloalkyl, aryl which can be substituted, or 3-indolyl.
机译:衍生物具有式I……,其中n为0、1或2,R为氢,烷基或芳烷基,R 1为氢或烷基,烯基,环烷基,环烯基,环烷基烷基,任选取代的芳基或R 2为可被取代的部分氢化的芳基,芳基-(C 1 -C 4)-烷基或芳酰基-C 1-烷基,它们均可被取代,单环或双环杂环基或天然氨基酸的侧链。氢,烷基,烯基或芳烷基,X是烷基,烯基,环烷基,可被取代的芳基或3-吲哚基。

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