首页> 外国专利> Pyrido (3,2,1-ij) -1,3,4-benzoxadiazina, process for their preparation, pharmaceutical preparations and corresponding intermediates used in the process.

Pyrido (3,2,1-ij) -1,3,4-benzoxadiazina, process for their preparation, pharmaceutical preparations and corresponding intermediates used in the process.

机译:Pyrido(3,2,1-ij)-1,3,4-benzoxadiazina,其制备方法,药物制剂和该方法中使用的相应中间体。

摘要

The invention relates to tricyclic compounds general formula (I), wherein R1 is a hydrogen atom or a protecting group carboxy, R2 is an atom of hydrogen or a lower alkyl substituted IF NECESSARY FOR A halogen atom , R3 and R4 are each independently a hydrogen atom or a radical lower alkyl substituted by a hydroxy group or an amino; X is a halogen atom; R5 and R6 are, independently of one another, a hydrogen atom or an alkyl radical CASE IF REPLACED BY A GROUP hydroxy, lower alkoxy group or an amino R5, R6 and R7 are as defined in the invention. Process for their preparation and pharmaceutical preparations containing them. FINISHED GOODS PRESENTED antibacterial activity.
机译:本发明涉及通式(I)的三环化合物,其中R 1是氢原子或保护基羧基,R 2是氢或被低级烷基取代的原子。如果对于卤素原子是必要的,R 3和R 4各自独立地是氢原子或被羟基或氨基取代的低级烷基的基团; X是卤素原子; R 5和R 6彼此独立地是氢原子或烷基,如果被基团取代,则羟基,低级烷氧基或氨基R 5,R 6和R 7如本发明中所定义。它们的制备方法和包含它们的药物制剂。成品具有抗菌活性。

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