首页> 外国专利> USE OF RE-DISPERSIBLE POLYMERIC POWDER OR POLYMERIC GRANULE FOR COATING AND PHARMACEUTICAL OR AGROCHEMICAL DOSAGE FORM

USE OF RE-DISPERSIBLE POLYMERIC POWDER OR POLYMERIC GRANULE FOR COATING AND PHARMACEUTICAL OR AGROCHEMICAL DOSAGE FORM

机译:将可再分散的聚合物粉末或聚合物颗粒用于涂料和药物或农用化学剂型

摘要

PROBLEM TO BE SOLVED: To obtain polymeric powder or polymeric granules comprising a water-insoluble polymer and a water-soluble polymer, completely re-dispersible, suitable for uniform coating of pharmaceutical or agrochemical dosage form and enabling the easily controllable release of active ingredient(s). SOLUTION: The re-dispersible polymeric powder or granules comprises (a) 10-95 wt.% of polyvinyl acetate, (b) 5-90 wt.% of an N-vinylpyrrolidone-contg. polymer, (c) 0-20 wt.% of another water-soluble or water-swellable substance and d) 0-20 wt.% of water-insoluble pulverizing agent, and in some cases, (e) other additive(s), so as to coat a pharmaceutical or agrochemical dosage form. The polymeric powder or granules ensures the controlled release of the active substance, epoxiconazole into soil for at least 6 months through a polyvinyl acetate/polyvinyl pyrrolidone coat.
机译:要解决的问题:要获得包含水不溶性聚合物和水溶性聚合物的聚合物粉末或聚合物颗粒,该聚合物粉末完全可再分散,适合于药物或农用化学剂型的均匀包衣,并且能够轻松控制活性成分的释放( s)。解决方案:可再分散的聚合物粉末或颗粒包含(a)10-95 wt。%的聚乙酸乙烯酯,(b)5-90 wt。%的N-乙烯基吡咯烷酮-浓缩物。聚合物;(c)0-20 wt。%的另一种水溶性或水溶胀性物质,和d)0-20 wt。%的水不溶性粉碎剂,在某些情况下,(e)其他添加剂,以制成药物或农药的剂型。聚合物粉末或颗粒可确保通过聚乙酸乙烯酯/聚乙烯吡咯烷酮涂层将活性物质epoxiconazole控释到土壤中至少6个月。

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